Compile Data Set for Download or QSAR
Report error Found 248 for UniProtKB: P05412
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50135483(1-(6-methoxy-2-(thiophen-2-yl)quinazolin-4-ylamino...)
Affinity DataIC50: 3nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50135482(1-(5-Methoxy-2-thiophen-2-yl-quinazolin-4-ylamino)...)
Affinity DataIC50: 8nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092879(2-Chloro-4-methyl-pyrimidine-5-carboxylic acid (3,...)
Affinity DataIC50: 20nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340608(8-(6-methylpyridin-3-yl)-N-(4-(3-morpholino-1H-1,2...)
Affinity DataIC50: 20nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090430(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 20nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092879(2-Chloro-4-methyl-pyrimidine-5-carboxylic acid (3,...)
Affinity DataIC50: 20nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50090430(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 20nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50295171(CHEMBL487194 | AILANTHINONE)
Affinity DataIC50: 32nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044568(CHEMBL85822)
Affinity DataIC50: 35nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50349194(NSC-14975 | GLAUCARUBINONE)
Affinity DataIC50: 40nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340606(N-(4-(3-(6-methylpyridin-3-yl)-1H-1,2,4-triazol-1-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340627(7,8-bis(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morpholi...)
Affinity DataIC50: 40nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340628(7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morpholino-1H...)
Affinity DataIC50: 40nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044567(CHEMBL86615)
Affinity DataIC50: 45nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340629(8-methoxy-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-mor...)
Affinity DataIC50: 50nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50062648(2-Chloro-4-trifluoromethyl-pyrimidine-5-carboxylic...)
Affinity DataIC50: 50nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50062648(2-Chloro-4-trifluoromethyl-pyrimidine-5-carboxylic...)
Affinity DataIC50: 50nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50213931(tylophorinidine | CHEMBL250854)
Affinity DataIC50: 65nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50213932([(R)-(+)-deoxytylophorinidine | CHEMBL250474)
Affinity DataIC50: 68nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50295170(6R-senecionylchaparrin | CHEMBL564009)
Affinity DataIC50: 71nMAssay Description:Inhibition of TPA-induced AP1 transfected in HEK293 cells assessed as inhibition of beta-lactamase reporter activity treated 1 hr before TPA stimulat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044564(CHEMBL315804)
Affinity DataIC50: 98nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044572(CHEMBL3341912)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090407(ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamin...)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090444(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340622(8-chloro-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morp...)
Affinity DataIC50: 100nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092877(2-Fluoro-4-trifluoromethyl-pyrimidine-5-carboxylic...)
Affinity DataIC50: 100nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092877(2-Fluoro-4-trifluoromethyl-pyrimidine-5-carboxylic...)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50090444(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 100nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50213934(tylophorinine | CHEMBL398325)
Affinity DataIC50: 110nMAssay Description:Inhibition of AP1-mediated gene transcription in HepG2 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340600(N-(4-(3-morpholino-1H-1,2,4-triazol-1-yl)phenyl)-7...)
Affinity DataIC50: 120nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340626(8-cyclopropyl-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3...)
Affinity DataIC50: 130nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50349194(NSC-14975 | GLAUCARUBINONE)
Affinity DataEC50:  130nMAssay Description:Inhibition of TPA-induced AP-1 activity expressed in human HEK293T cells treated 1 hr before TPA challenge measured after 18 hrs by FRET based beta-l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50349193(CHEMBL1807644)
Affinity DataEC50:  130nMAssay Description:Inhibition of AP-1 (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340624(8-methyl-7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-morp...)
Affinity DataIC50: 160nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090443(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090420(4-(3-Methyl-2,5-dioxo-2,5-dihydro-pyrrol-1-ylamino...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092882(2,4-Dichloro-pyrimidine-5-carboxylic acid (3,5-bis...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090406(1-[5-(4,5-Dihydro-oxazol-2-yl)-2-thiophen-2-yl-pyr...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090431(3-methyl-1-(5-(4-methyloxazol-2-yl)-2-(thiophen-2-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340614(N-(4-(3-methyl-1H-1,2,4-triazol-1-yl)phenyl)-8-(th...)
Affinity DataIC50: 200nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090442(3-methyl-1-(5-(2-methyl-2H-tetrazol-5-yl)-2-(thiop...)
Affinity DataIC50: 200nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092882(2,4-Dichloro-pyrimidine-5-carboxylic acid (3,5-bis...)
Affinity DataIC50: 200nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044566(CHEMBL87274)
Affinity DataIC50: 210nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340610(8-(3-fluoro-4-methoxyphenyl)-N-(4-(3-morpholino-1H...)
Affinity DataIC50: 250nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50340607(7-(1-methyl-1H-pyrazol-4-yl)-N-(4-(3-(pyridin-2-yl...)
Affinity DataIC50: 290nMAssay Description:Inhibition of c-JunMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090450(3-methyl-1-(5-(5-methyl-1,3,4-oxadiazol-2-yl)-2-(t...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090435(3-methyl-1-(5-(3-methylisoxazol-5-yl)-2-(thiophen-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetProtein c-Fos/Transcription factor Jun(Human)
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50090449(ethyl 2-(4-chlorophenyl)-4-(3-methyl-2,5-dioxo-2H-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1 (activator protein-1) mediated transcriptional activation in Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50044570(CHEMBL87433)
Affinity DataIC50: 300nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
University of Texas Medical Branch

Curated by ChEMBL
LigandPNGBDBM50092890(2-Chloro-pyrimidine-5-carboxylic acid (3,5-bis-tri...)
Affinity DataIC50: 300nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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