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Report error Found 31 of affinity data for UniProtKB/TrEMBL: P08151
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378034BDBM50378034(NSC-287088 | PHYSALIN B | CHEMBL504404)
Affinity DataIC50: 600nMAssay Description:Inhibition of GLI1 (unknown origin) transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378034BDBM50378034(NSC-287088 | PHYSALIN B | CHEMBL504404)
Affinity DataIC50: 620nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378033BDBM50378033(PHYSALIN F)
Affinity DataIC50: 660nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50612863BDBM50612863(CHEMBL5281322)
Affinity DataIC50: 700nMAssay Description:Inhibition of GLI1 (unknown origin) transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50557557BDBM50557557(CHEMBL504910)
Affinity DataIC50: 700nMAssay Description:Inhibition of GLI1 (unknown origin) transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321859BDBM50321859(2-(3-Benzoylphenyl)-N-(1H-indol-5-yl)-N-propylprop...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human Gli1 expressed in mouse C3H10T1/2 cells assessed as inhibition of transcriptional activity after 24 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2581BDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240978BDBM50240978(5,6-dihydroxy-8,9-dihydro-1H-indolo[2,3-a]pyrrolo[...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240682BDBM50240682(2,10-dihydroxy-6,7,12,13-tetrahydro-5H-indolo[2,3-...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240964BDBM50240964(2-hydroxy-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50321858BDBM50321858(2-(3-Benzoylphenyl)-N-(1H-indol-6-yl)-N-propylprop...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human Gli1 expressed in mouse C3H10T1/2 cells assessed as inhibition of transcriptional activity after 24 hrs by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50612864BDBM50612864(CHEMBL5280113)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of GLI1 (unknown origin) transcriptional activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607892BDBM50607892(CHEBI:3914 | (+)-Crinamine | CHEMBL516991)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of GLI1-mediated transcriptional activity in human HaCaT cells coexpressing luciferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293859BDBM50293859((S)-2-(3-Benzoylphenyl)-N-(4-hydroxyphenethyl)-N-p...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of exogenously transfected human Gli1-mediated transcriptional activity in mouse C3H10T1/2 cells after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50241296BDBM50241296(Zerumbone | CHEMBL245412)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293858BDBM50293858((S)-2-(3-Benzoylphenyl)-N,N-bis(4-hydroxyphenethyl...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of exogenously transfected human Gli1-mediated transcriptional activity in mouse C3H10T1/2 cells after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534830BDBM50534830(CHEMBL4453685)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Shh-N-induced Gli1 (unknown origin) expressed in mouse Shh Light2 cells assessed as Gli1-mediated mediated transcription incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293861BDBM50293861((S)-2-(3-Benzoylphenyl)-N-(4-hydroxyphenethyl)prop...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of exogenously transfected human Gli1-mediated transcriptional activity in mouse C3H10T1/2 cells after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50293860BDBM50293860((S)-2-(3-Benzoylphenyl)-N-(3,4-dihydroxyphenethyl)...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of exogenously transfected human Gli1-mediated transcriptional activity in mouse C3H10T1/2 cells after 24 hrs by luciferase reporter gene ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50612862BDBM50612862(CHEMBL5271777)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of GLI1-mediated transcriptional activity in human HaCaT cells coexpressing luciferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50221066BDBM50221066(9,10-(methylenedioxy)-3,12-didehydrogalanthan-1alp...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of GLI1-mediated transcriptional activity in human HaCaT cells coexpressing luciferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50534831BDBM50534831(CHEMBL4435840)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Shh-N-induced Gli1 (unknown origin) expressed in mouse Shh Light2 cells assessed as Gli1-mediated mediated transcription incubated for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 23208BDBM23208(cid_64971 | CHEMBL269277 | (1R,2R,5S,8R,9R,10R,13R...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 23208BDBM23208(cid_64971 | CHEMBL269277 | (1R,2R,5S,8R,9R,10R,13R...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of GLI1-mediated transcriptional activity in human HaCaT cells by luciferase based reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249140BDBM50249140(colubrinic acid | CHEMBL470503)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249140BDBM50249140(colubrinic acid | CHEMBL470503)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of GLI1-mediated transcriptional activity in human HaCaT cells by luciferase based reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249557BDBM50249557(2-((3-(2-(dimethylamino)benzyl)-2-(pyridin-4-yl)-t...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human Gli1-mediated transcriptional activity in human Rh30 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/31/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249188BDBM50249188(Alphitolic acid | CHEMBL511805)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of Gli1-mediated transcription expressed in human PANC1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249188BDBM50249188(Alphitolic acid | CHEMBL511805)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of GLI1-mediated transcriptional activity in human HaCaT cells by luciferase based reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50274058BDBM50274058(ceanothanolic acid | CHEMBL522108)
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of GLI1-mediated transcriptional activity in human HaCaT cells by luciferase based reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed
TargetZinc finger protein GLI1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50377959BDBM50377959(CHEMBL491069)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of GLI1-mediated transcriptional activity in human HaCaT cells by luciferase based reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed