Compile Data Set for Download or QSAR
Report error Found 128 of affinity data for UniProtKB/TrEMBL: P19367
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  5.5nMAssay Description:Binding affinity to human HK1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169033(CHEMBL3806069)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169038(CHEMBL3804841)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169026(CHEMBL3805148)
Affinity DataIC50: 16nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169032(CHEMBL3805398)
Affinity DataIC50: 20nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169037(CHEMBL3805205)
Affinity DataIC50: 20nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169034(CHEMBL3805734)
Affinity DataIC50: 25nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169031(CHEMBL3805905)
Affinity DataIC50: 32nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169017(CHEMBL3804930)
Affinity DataIC50: 40nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169028(CHEMBL3805598)
Affinity DataIC50: 160nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169023(CHEMBL3805753)
Affinity DataIC50: 160nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169015(CHEMBL3805460)
Affinity DataIC50: 790nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169042(CHEMBL3806103)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80810(cid_240739 | 7-azanyl-6-chloranyl-5,8-bis(oxidanyl...)
Affinity DataEC50:  1.06E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169036(CHEMBL3806028)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169013(CHEMBL3805703)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169019(CHEMBL3805765)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169039(CHEMBL3806132)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169025(CHEMBL3806250)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169041(CHEMBL3805653)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80825(MLS002701915 | cid_45479889 | SMR001565499 | 7,10-...)
Affinity DataEC50:  5.20E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM52656(MLS000681605 | 1-[5-acetyl-3-methyl-6-(3-nitrophen...)
Affinity DataEC50:  6.54E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50673(cid_4834997 | N-[4-[2-[(4-morpholin-4-ylsulfonylph...)
Affinity DataEC50:  7.65E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80766(SMR000048155 | methyl 2-(7-fluoranyl-2-methyl-[1,3...)
Affinity DataEC50:  8.10E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM63324(3-[[5-(4-ethylphenyl)-6H-1,3,4-thiadiazin-2-yl]ami...)
Affinity DataEC50:  8.26E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169040(CHEMBL3804874)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM45724(SMR000414744 | 4-[(3-chloro-1,4-dioxonaphthalen-2-...)
Affinity DataEC50:  1.06E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80808(MLS002477170 | 2-(2-azanyl-6-methylsulfanyl-purin-...)
Affinity DataEC50:  1.18E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169014(CHEMBL3806183)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM42405(N-(2-piperazin-1-yl-1,2-dihydroacenaphthylen-1-yl)...)
Affinity DataEC50:  1.36E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80809(3-[1-methyl-5-[(1-methyl-5-pyridin-3-yl-pyrrol-2-y...)
Affinity DataEC50:  1.42E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80788(SMR000253852 | ethyl (5E)-5-[2-[(2-methoxyphenyl)a...)
Affinity DataEC50:  1.53E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80784(SMR000236766 | cid_2135781 | MLS000722098 | 2-[[5-...)
Affinity DataEC50:  1.63E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80798(3-[[5-(2,4-dimethoxyphenyl)-6H-1,3,4-thiadiazin-2-...)
Affinity DataEC50:  1.74E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80796(MLS000772545 | SMR000377243 | cid_5026871 | N-(4-f...)
Affinity DataEC50:  1.78E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80806(3-[1,3-bis(oxidanylidene)benzo[de]isoquinolin-2-yl...)
Affinity DataEC50:  1.79E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80781(MLS000335157 | (5E)-5-(2-anilino-4H-1,3,4-thiadiaz...)
Affinity DataEC50:  1.82E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM63662(cid_3032310 | 1,3-dihydroindole-2-thione | SMR0003...)
Affinity DataEC50:  1.93E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM50169043(CHEMBL3806095)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2017
Entry Details Article
PubMed
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80799(SMR000364573 | MLS000774989 | cid_4883712 | 3-[[5-...)
Affinity DataEC50:  2.01E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM52665(SMR000312275 | MLS000681598 | cid_5295671 | 1-(5-e...)
Affinity DataEC50:  2.08E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80785(SMR000254526 | ethyl (5E)-5-[2-[(4-ethoxyphenyl)am...)
Affinity DataEC50:  2.11E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80804(MLS001198575 | 2-ethyl-3-methyl-1-(methylamino)-4-...)
Affinity DataEC50:  2.11E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80768(MLS000118337 | cid_5309702 | 1-[2-(azepan-1-yl)-2-...)
Affinity DataEC50:  2.17E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80774(MLS000566795 | SMR000153752 | 5-(2,3-dihydro-1,4-b...)
Affinity DataEC50:  2.39E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80764(N-{2-[4-(2-Hydroxy-ethyl)-piperazin-1-yl]-acenapht...)
Affinity DataEC50:  2.40E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80779(SMR000172259 | cid_2913537 | N-[2-(4-Methyl-4H-[1,...)
Affinity DataEC50:  2.47E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80786(MLS000390436 | SMR000255403 | cid_8968424 | 5-(2,5...)
Affinity DataEC50:  2.89E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM66618(MLS000830340 | N-[2-(4-acetylpiperazin-1-yl)-1,2-d...)
Affinity DataEC50:  2.94E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetHexokinase-1(Human)TBA
LigandPNGBDBM80795(SMR000370724 | cid_4286294 | MLS001002761 | 5-[2,5...)
Affinity DataEC50:  2.95E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
Displayed 1 to 50 (of 128 total ) | Next | Last >>
Jump to: