Compile Data Set for Download or QSAR
Report error Found 1369 for UniProtKB: P30994
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608949BDBM50608949(CHEMBL5270056)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001778BDBM50001778((Lu 23-086)1-(2-{4-[1-(4-Fluoro-phenyl)-1H-indol-3...)
Affinity DataIC50: 0.0820nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069019BDBM50069019(7-Chloro-1-(4-fluoro-phenyl)-8,9-dimethoxy-4-methy...)
Affinity DataKi:  0.0900nMAssay Description:Affinity for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218398BDBM50218398(CHEMBL1907861)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004819BDBM50004819(CHEMBL135917 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.0960nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010041BDBM50010041(CHEMBL84087 | {1-[3-(1,1-Dioxo-1H-1lambda*6*-napht...)
Affinity DataIC50: 0.100nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608952BDBM50608952(CHEMBL5279881)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608953BDBM50608953(CHEMBL5284094)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608950BDBM50608950(CHEMBL5280131)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608951BDBM50608951(CHEMBL5277645)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004807BDBM50004807(CHEMBL334349 | 8-[4-(4-Fluoro-phenyl)-4-oxo-butyl]...)
Affinity DataKi:  0.130nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218392BDBM50218392(CHEMBL79277)
Affinity DataKi:  0.140nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50025124BDBM50025124(3-{2-[4-(4-Fluoro-benzoyl)-piperidin-1-yl]-ethyl}-...)
Affinity DataKi:  0.170nMAssay Description:Evaluated for binding activity against [3H]ketanserin as radioligand for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608956BDBM50608956(CHEMBL94655)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001885BDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  0.200nMAssay Description:Affinity for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50407849BDBM50407849(CHEMBL96480)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608955BDBM50608955(CHEMBL96427)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010048BDBM50010048(CHEMBL418929 | 2-[3-(4-Phenyl-piperidin-1-yl)-prop...)
Affinity DataIC50: 0.200nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001885BDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  0.200nMAssay Description:The binding affinity was measured on 5-hydroxytryptamine 2 receptor in rat brain tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50407853BDBM50407853(CHEMBL94644)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 85862BDBM85862(1-(2-Chloro-3,4-dimethoxybenzyl)-6-methyl-2,3,4,9-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001991BDBM50001991(CHEMBL275496 | 1-(2-{4-[5-Chloro-1-(4-fluoro-pheny...)
Affinity DataIC50: 0.240nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218396BDBM50218396(CHEMBL315259)
Affinity DataKi:  0.240nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010044BDBM50010044(FANANSERIN | ChEMBL_131689 | 2-{3-[4-(4-Fluoro-phe...)
Affinity DataKi:  0.260nMAssay Description:Binding constant against 5-hydroxytryptamine 2 receptor (in vivo)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010044BDBM50010044(FANANSERIN | ChEMBL_131689 | 2-{3-[4-(4-Fluoro-phe...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity to rat cerebral cortex homogenate 5-HT2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001775BDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataKi:  0.260nMAssay Description:The compound was tested for its binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [3H]ketanserin radioligand in rat cerebral cort...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010049BDBM50010049(CHEMBL79375 | 4-{4-[3-(1,1-Dioxo-1H-1lambda*6*-nap...)
Affinity DataIC50: 0.300nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002008BDBM50002008(CHEMBL267304 | 1-(2-{4-[1-(4-Fluoro-phenyl)-5-meth...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001990BDBM50001990(CHEMBL273516 | 5-Chloro-1-(4-fluoro-phenyl)-3-(4-m...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of [3H]ketanserin binding to dopamine 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 30704BDBM30704(METERGOLINE | (phenylmethyl) N-[[(6aR,9S,10aR)-4,7...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 (5-HT2) receptor using [3H]KET as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50024205BDBM50024205(CHEMBL18331 | 3-{2-[4-(4-Fluoro-benzoyl)-piperidin...)
Affinity DataKi:  0.300nMAssay Description:Evaluated for the binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 receptor binding site by using [3H]- KET as a radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004818BDBM50004818(CHEMBL136942 | 3-Ethyl-8-[4-(4-fluoro-phenyl)-4-ox...)
Affinity DataKi:  0.310nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218397BDBM50218397(CHEMBL83611)
Affinity DataKi:  0.320nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001786BDBM50001786(1-[2-[4-[5-chloro-1-(4-fluorophenyl)-indol-3-yl]-1...)
Affinity DataIC50: 0.390nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor from rat cortical membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064708BDBM50064708((R)-2-(4-Bromo-2,5-dimethoxy-phenyl)-1-methyl-ethy...)
Affinity DataKi:  0.390nMAssay Description:Affinity towards [3H]- DOB -labeled 5-hydroxytryptamine 2 receptor sites in rat cortical homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001786BDBM50001786(1-[2-[4-[5-chloro-1-(4-fluorophenyl)-indol-3-yl]-1...)
Affinity DataIC50: 0.390nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001775BDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataIC50: 0.400nMAssay Description:Compound was tested for the displacement of [3H]ketanserin from serotonin 5-hydroxytryptamine 2 receptor from rat cortical membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21395BDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  0.400nMAssay Description:Evaluated for the binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 receptor binding site by using [3H]- KET as a radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010038BDBM50010038(CHEMBL79927 | 2-[3-(4-Benzo[d]isothiazol-3-yl-pipe...)
Affinity DataIC50: 0.400nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001775BDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50064708BDBM50064708((R)-2-(4-Bromo-2,5-dimethoxy-phenyl)-1-methyl-ethy...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 receptor binding site by using [3H]- DOB as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007692BDBM50007692(TIOSPERONE | CHEMBL35057 | CHEMBL1204189 | 8-[4-(4...)
Affinity DataIC50: 0.400nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor measured using radioligand ([3H]spiperone) binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001775BDBM50001775(cid_5074 | Ritanserine | 6-(2-{4-[Bis-(4-fluoro-ph...)
Affinity DataIC50: 0.400nMAssay Description:Compound was tested for the displacement of [3H]ketanserin from serotonin 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Rat)
Univ. Grenoble Alpes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50608954BDBM50608954(CHEMBL329479)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]-ketanserin from rat 5-HT2B expressed in mouse NIH/3T3 cells assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50069011BDBM50069011(1-(4-Fluoro-phenyl)-8,9-dimethoxy-4-methyl-2,2a,3,...)
Affinity DataKi:  0.410nMAssay Description:Affinity for 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004805BDBM50004805(CHEMBL136852 | 3-Butyl-8-[4-(4-fluoro-phenyl)-4-ox...)
Affinity DataKi:  0.410nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21395BDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKd:  0.420nMAssay Description:Binding affinity for membrane-bound 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50218399BDBM50218399(CHEMBL79643)
Affinity DataKi:  0.440nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/1/2012
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21397BDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  0.450nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
H. Lundbeck

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002001BDBM50002001(CHEMBL269679 | 1-(2-{4-[5-Fluoro-1-(4-fluoro-pheny...)
Affinity DataIC50: 0.480nMAssay Description:Inhibition of [3H]ketanserin binding to rat 5-hydroxytryptamine 2 receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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