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TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422795(CHEMBL202585)
Affinity DataIC50: 0.00100nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50059997(7 beta-Spirobenzocyclohexylnaltrexone | CHEMBL1016...)
Affinity DataKi:  0.00190nMAssay Description:Inhibition of [3H]-NTI binding to Opioid receptor delta 1 from mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422811(CHEMBL204716)
Affinity DataIC50: 0.00200nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50059994(7 alpha-Spirobenzocyclohexylnaltrexone | CHEMBL105...)
Affinity DataKi:  0.00410nMAssay Description:Inhibition of [3H]-NTI binding to Opioid receptor delta 1 from mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422791(CHEMBL204480)
Affinity DataIC50: 0.00500nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetDelta-type/Mu-type opioid receptor(Mouse)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50376594(CHEMBL260120)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse frontal cortex assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50121648(2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...)
Affinity DataIC50: 0.0150nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50043724(CHEMBL339320 | (S)-2-({(4R,7S)-13-[(S)-2-Amino-3-(...)
Affinity DataIC50: 0.0160nMAssay Description:Inhibitory potency against Opioid receptor delta 1 was determined in electrically induced smooth muscle contractions of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50061295((S)-2-{[(4R,7S,13S)-13-[(S)-2-Amino-3-(4-hydroxy-p...)
Affinity DataIC50: 0.0160nMAssay Description:Inhibitory potency against Opioid receptor delta 1 was determined in electrically induced smooth muscle contractions of mouse vas deferens (MVD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50142622(CHEMBL3758292)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at delta-opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2017
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422809(CHEMBL204136)
Affinity DataIC50: 0.0200nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50111905((S)-4-[(S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 0.0220nMAssay Description:In vitro biological activity by electrically induced smooth muscle contractions in mouse vas deferens (Opioid receptor delta 1); inhibitory concentra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50121645(2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)pr...)
Affinity DataIC50: 0.0260nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50121645(2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)pr...)
Affinity DataIC50: 0.0260nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50043721((S)-2-{[(4R,7S)-13-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 0.0280nMAssay Description:Inhibitory concentration against delta opioid receptor of electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50058154(7-(4'-Methoxy-2'-spiroindanyl)naltrexone | CHEMBL2...)
Affinity DataKi:  0.0280nMAssay Description:The compound tested for agonistic activity against Opioid receptor delta 1 using [3H]- NT1 as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50334989((R)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataIC50: 0.0290nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164 | US12215173, Compound Naltrindole)
Affinity DataKi:  0.0300nMAssay Description:Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on delta-opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDelta-type/Mu-type opioid receptor(Mouse)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50554766(CHEMBL4795492)
Affinity DataEC50:  0.0316nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type/Mu-type opioid receptor(Mouse)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50554766(CHEMBL4795492)
Affinity DataEC50:  0.0320nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179191(H-Dmt-Tic-NH-CH2-Bid | 2-[2-Amino-3-(4-hydroxy-2,6...)
Affinity DataIC50: 0.0350nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179191(H-Dmt-Tic-NH-CH2-Bid | 2-[2-Amino-3-(4-hydroxy-2,6...)
Affinity DataIC50: 0.0350nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422804(CHEMBL202578)
Affinity DataIC50: 0.0400nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity against Opioid receptor delta 1 receptor binding in ICR mouse brain membranes using the radioligand [3H]naltrindoleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001462(CHEMBL124435 | 3-[(2-{2-[2-Amino-3-(4-hydroxy-phen...)
Affinity DataIC50: 0.0803nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50391602(CHEMBL2147915)
Affinity DataKi:  0.0920nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50253136(CHEMBL4075409)
Affinity DataKi:  0.109nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2019
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory activity against Mouse vas deferens smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataIC50: 0.115nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50272169(UFP-512 | H-Dmt-Tic-NH-(S)CH(CH2-COOH)-Bid | (S)-3...)
Affinity DataIC50: 0.120nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50272169(UFP-512 | H-Dmt-Tic-NH-(S)CH(CH2-COOH)-Bid | (S)-3...)
Affinity DataIC50: 0.120nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50360146(CHEMBL1929368)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50297288((S)-4-(1H-benzo[d]imidazol-2-yloxy)-3-((S)-2-((S)-...)
Affinity DataIC50: 0.120nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50060065(2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataKd:  0.126nMAssay Description:Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50422803(CHEMBL382024)
Affinity DataIC50: 0.126nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50179191(H-Dmt-Tic-NH-CH2-Bid | 2-[2-Amino-3-(4-hydroxy-2,6...)
Affinity DataIC50: 0.130nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50010532(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50: 0.130nMAssay Description:Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50027229(CHEMBL2375157)
Affinity DataIC50: 0.130nMAssay Description:Agonist activity at delta opioid receptor by mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50297286(1H-benzo[d]imidazol-2-yl 2-((S)-2-((S)-2-amino-3-(...)
Affinity DataIC50: 0.130nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50294428(SN-28 | CHEMBL552308)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50329100(CHEMBL1270475)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50009142(3-[1-[1-[1-amino-2-(4-hydroxyphenyl)-(1S)-ethylcar...)
Affinity DataIC50: 0.140nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50494888(CHEMBL4296733)
Affinity DataKi:  0.141nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellum after 1 hr by liquid scintillation counting a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50391591(CHEMBL2147904)
Affinity DataKi:  0.143nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50329100(CHEMBL1270475)
Affinity DataKi:  0.143nMAssay Description:Displacement of [3H]-DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellum after 1 hr by liquid scintillation counting a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50391594(CHEMBL2147907)
Affinity DataKi:  0.146nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50001468(deltorphin C | CHEMBL317956 | H-Tyr-D-Ala-Phe-Asp-...)
Affinity DataIC50: 0.147nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50009146(CHEMBL26575 | (S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(...)
Affinity DataIC50: 0.147nMAssay Description:Agonist activity at delta-opioid receptor in mouse vasa deferens assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2020
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50391595(CHEMBL2147908)
Affinity DataKi:  0.148nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50491882(CHEMBL3215908)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed
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