Compile Data Set for Download or QSAR
Report error Found 88 of affinity data for UniProtKB/TrEMBL: P51577
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50029031(CHEMBL223344 | 1-Amino-4-{4-[4-chloro-6-(3-sulfo-p...)
Affinity DataKi:  46.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50422739(CHEMBL413145)
Affinity DataIC50: 81nMAssay Description:Inhibitory concentration against rat P2X purinoceptor 1 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50300129(CHEMBL572528 | Cibacron Blue 3Ga | CIBACRON BLUE)
Affinity DataKi:  128nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50: 233nMAssay Description:Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85044(NSC_8272 | CAS_8272 | CAS_115-39-9 | Bromphenol bl...)
Affinity DataKi:  302nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50000029(suramin | SURAMIN HEXASODIUM | CHEMBL265502 | 4-Me...)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85043(CHEMBL69234 | CAS_149017-66-3 | NSC_6093163 | PPAD...)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50399207(CHEMBL2180179)
Affinity DataIC50: 750nMAssay Description:Antagonist activity at rat P2X4R expressed in HEK293 cells preincubated for 2 mins followed by ATP addition and measured after 4 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50399183(CHEMBL2180160)
Affinity DataIC50: 928nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  1.00E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  1.00E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50118234(MRS 2160 | CHEMBL129904)
Affinity DataKd:  1.60E+3nMAssay Description:Dissociation constant of the compound at P2X purinoceptor 1 (P2X1) from rat vas deferens was reportedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50399165(CHEMBL2180137)
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50118217(PHOSPHOTHIOPHOSPHORIC ACID-ADENYLATE ESTER | ATPga...)
Affinity DataEC50:  2.30E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataIC50: 2.45E+3nMAssay Description:Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 10 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataIC50: 2.45E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85043(CHEMBL69234 | CAS_149017-66-3 | NSC_6093163 | PPAD...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of inward ion current elicited by ATP at rat P2X4 receptor (mutant type)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50399190(CHEMBL2180149)
Affinity DataIC50: 4.04E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50370141(TNP-ATP)
Affinity DataIC50: 4.71E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50399166(CHEMBL2180136)
Affinity DataIC50: 6.08E+3nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50118232(ATP, 2-meS | CHEMBL336208 | 2-MeSATP)
Affinity DataEC50:  7.40E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50118234(MRS 2160 | CHEMBL129904)
Affinity DataIC50: 9.60E+3nMAssay Description:The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) receptor from rat vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268966(Sodium 1-Amino-4-[4-([1,3]diazine-2-ylamino)phenyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268876(Disodium 1-amino-4-[4-(4-chloro-6-methoxy-[1,3,5]t...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336782(Sodium 1-Amino-4-[4-(4,6-dihydroxy[1,3,5]triazine-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50118229(MRS 2179 | CHEMBL129841)
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM, expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50118232(ATP, 2-meS | CHEMBL336208 | 2-MeSATP)
Affinity DataEC50:  1.00E+4nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50399164(CHEMBL2180138)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336785(sodium 1-amino-4-(cyclohexylamino)-9,10-dioxo-9,10...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268574(Sodium 1-amino-4-[1-naphthylamino]-9,10-dioxo-9,10...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336786(sodium 1-amino-9,10-dioxo-4-(o-tolylamino)-9,10-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336787(sodium 1-amino-9,10-dioxo-4-(m-tolylamino)-9,10-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336788(sodium 1-amino-9,10-dioxo-4-(p-tolylamino)-9,10-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336791(sodium 1-amino-4-(2,3-dimethylphenylamino)-9,10-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336792(sodium 1-amino-4-(2,4-dimethylphenylamino)-9,10-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268687(sodium 1-amino-4-(2-hydroxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50227032(acid blue 25 | sodium 1-amino-9,10-dioxo-4-(phenyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336783(1-amino-2-methyl-4-(phenylamino)anthracene-9,10-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336784(1-amino-2-methyl-4-(m-tolylamino)anthracene-9,10-d...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336773(sodium 1-amino-9,10-dioxo-4-(2-sulfonatophenylamin...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268686(sodium 1-amino-9,10-dioxo-4-(4-sulfophenylamino)-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268685(sodium 1-amino-4-(2-carboxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336774(sodium 1-amino-4-(3-carboxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336775(sodium 1-amino-4-(4-carboxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268635(sodium 1-amino-4-(2-aminophenylamino)-9,10-dioxo-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336776(sodium 1-amino-4-(3-aminophenylamino)-9,10-dioxo-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268636(Sodium 1-Amino-4-(4-aminophenylamino)-9,10-dioxo-9...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50268725(sodium 1-amino-4-(4-hydroxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336767(PSB-716 | sodium 1-amino-4-(2-methoxyphenylamino)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Max-Planck Institute For Experimental Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50336768(sodium 1-amino-4-(3-methoxyphenylamino)-9,10-dioxo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against rat P2X4 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2013
Entry Details Article
PubMed
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