TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair
TargetInterferon-induced, double-stranded RNA-activated protein kinase /Eukaryotic translation initiation factor 2-alpha kinase 3 [536-1116]/Small ubiquitin-related modifier 1/eIF-2-alpha kinase GCN2 (Human)
Hibercell
US Patent
Hibercell
US Patent
Affinity DataIC50: 25nMAssay Description:In vitro Inhibition of PERK Enzyme Activity (isolated) Recombinant human EIF2AK2 (PKR) catalytic domain (amino acids 252-551), EIF2AK3 (PERK) catalyt...More data for this Ligand-Target Pair

















































