TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 28nM Kd: 5.30E+3nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 5.70E+3nM Kd: 160nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 4.10E+4nM Kd: 4.90E+3nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 4.10E+4nM Kd: 6.00E+3nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: 8.00E+3nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 3.50E+4nM Kd: 9.30E+3nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.00E+5nM Kd: 1.00E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 6.50E+4nM Kd: 1.20E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 4.90E+4nM Kd: 1.60E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKi: 3.10E+4nM ΔG°: -25.5kJ/moleT: 2°CAssay Description:Reactions were performed in duplicate at 22 C in 50 mM NaH2PO4 buffer (pH 7) with 20 nM enzyme and 20 mM fresh sodium dithionite. Small molecules wer...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: >3.30E+4nMAssay Description:To access the ability of compounds to inhibit the catalytic activity of UGM, an HPLC assay was employed. Inhibition constants were determined by mon...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: 3.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UGM expressed in Escherichia coli BL21(DE3) assessed as dissociation constant by fluorescence polarization a...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 3.53E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 5.34E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 5.62E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 5.85E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: 6.30E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UGM expressed in Escherichia coli BL21(DE3) assessed as dissociation constant by fluorescence polarization a...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 6.43E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 8.27E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 9.47E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: 1.05E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UGM expressed in Escherichia coli BL21(DE3) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.46E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.49E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of His6-tagged Mycobacterium tuberculosis reduced UDP-galactopyranose mutase expressed in Escherichia coli BL21 assessed as reduction in U...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.65E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.68E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.84E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 1.84E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataKd: 1.97E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UGM expressed in Escherichia coli BL21(DE3) assessed as dissociation constant by fluorescence polarization a...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 2.05E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 2.09E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 2.25E+5nMAssay Description:Inhibition of His6-tagged Mycobacterium tuberculosis reduced UDP-galactopyranose mutase expressed in Escherichia coli BL21 assessed as reduction in U...More data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 2.27E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 2.45E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 2.59E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
TargetUDP-galactopyranose mutase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Wisconsin-Madison
University of Wisconsin-Madison
Affinity DataIC50: 2.64E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis UDP-galactose mutase expressed in Escherichia coli UDP-6 [3H]- GalfMore data for this Ligand-Target Pair
















































