Compile Data Set for Download or QSAR
Report error Found 3291 of affinity data for UniProtKB/TrEMBL: Q05397
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50513279BDBM50513279(CHEMBL4554455)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of human recombinant N-terminal His-tagged FAK (393 to 698 residues) expressed in baculovirus infected Sf9 insect cells using Poly (4:1 Gl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590475BDBM50590475(CHEMBL5170906)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590490BDBM50590490(CHEMBL5198068)
Affinity DataIC50: 0.108nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590479BDBM50590479(CHEMBL5196177)
Affinity DataIC50: 0.117nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590489BDBM50590489(CHEMBL5176233)
Affinity DataIC50: 0.124nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590488BDBM50590488(CHEMBL5206909)
Affinity DataIC50: 0.153nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590483BDBM50590483(CHEMBL5187385)
Affinity DataIC50: 0.161nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590484BDBM50590484(CHEMBL5190968)
Affinity DataIC50: 0.192nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590485BDBM50590485(CHEMBL5177776)
Affinity DataIC50: 0.194nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590474BDBM50590474(CHEMBL5176990)
Affinity DataIC50: 0.213nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554439BDBM50554439(CHEMBL4752642)
Affinity DataKi:  0.230nMAssay Description:Covalent inhibition of recombinant human N-terminal His-tagged FAK (393 to 698 residues) expressed in baculovirus infected Sf9 insect cells using Pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590477BDBM50590477(CHEMBL5204729)
Affinity DataIC50: 0.275nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590482BDBM50590482(CHEMBL5186801)
Affinity DataIC50: 0.296nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 155552BDBM155552(US9012461, 28)
Affinity DataIC50: 0.300nMpH: 7.4Assay Description:A biotin labeled peptide is used as substrate (amino acid sequence: Biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2)1S...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2015
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590487BDBM50590487(CHEMBL5199835)
Affinity DataIC50: 0.315nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590476BDBM50590476(CHEMBL5178369)
Affinity DataIC50: 0.315nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418652BDBM418652(4-{[4-({3- [methyl(methylsulfonyl)amino]benzyl} am...)
Affinity DataIC50: 0.380nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 155547BDBM155547(US9012461, 23)
Affinity DataIC50: 0.390nMpH: 7.4Assay Description:A biotin labeled peptide is used as substrate (amino acid sequence: Biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2)1S...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2015
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 755771BDBM755771(US20250214967, Compound A6)
Affinity DataIC50: 0.390nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 755769BDBM755769(N-(1-((1-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoiso...)
Affinity DataIC50: 0.400nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554449BDBM50554449(CHEMBL4750273)
Affinity DataKi:  0.400nMAssay Description:Covalent inhibition of recombinant human N-terminal His-tagged FAK (393 to 698 residues) expressed in baculovirus infected Sf9 insect cells using Pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50568532BDBM50568532(CHEMBL4742157)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50568532BDBM50568532(CHEMBL4742157)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 155545BDBM155545(US9012461, 21)
Affinity DataKd:  0.440nMpH: 7.4 T: 2°CAssay Description:Binding parameters of compounds were determined using a Biacore S51 sensor. An anti-GST antibody was immobilized onto a CM5 chip by primary amine-cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2015
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 155537BDBM155537(US9012461, 13)
Affinity DataKd:  0.470nMpH: 7.4 T: 2°CAssay Description:Binding parameters of compounds were determined using a Biacore S51 sensor. An anti-GST antibody was immobilized onto a CM5 chip by primary amine-cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2015
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50554448BDBM50554448(CHEMBL4783568)
Affinity DataKi:  0.470nMAssay Description:Covalent inhibition of recombinant human N-terminal His-tagged FAK (393 to 698 residues) expressed in baculovirus infected Sf9 insect cells using Pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 755772BDBM755772(US20250214967, Compound A7)
Affinity DataIC50: 0.470nMAssay Description:The inhibitory activity of a compound against FAK was determined in a buffer containing 5 mM HEPES, pH 7.5, 0.01% Triton, 0.5 mM EGTA, and 0.01% BRIJ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 155560BDBM155560(US9012461, 36)
Affinity DataKd:  0.480nMpH: 7.4 T: 2°CAssay Description:Binding parameters of compounds were determined using a Biacore S51 sensor. An anti-GST antibody was immobilized onto a CM5 chip by primary amine-cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2015
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 155525BDBM155525(US9012461, 1)
Affinity DataKd:  0.490nMpH: 7.4 T: 2°CAssay Description:Binding parameters of compounds were determined using a Biacore S51 sensor. An anti-GST antibody was immobilized onto a CM5 chip by primary amine-cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2015
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 418817BDBM418817(US10450297, Example 317 | US10450297, Example 318 ...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant FAK (unknown origin) by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50246239BDBM50246239(N-methyl-N-(2-((2-(1-oxoisoindolin-5-ylamino)-5-(t...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged FAK assessed as inhibition of poly-Glu-Tyr phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50207359BDBM50207359(CHEMBL3892377)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50592745BDBM50592745(CHEMBL5188373)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50207351BDBM50207351(CHEMBL3965256)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of NH2-terminal His6-tagged FAK kinase domain (410 to 689 residues) (unknown origin) expressed in baculovirus infected sf9 cells using p(G...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2018
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590486BDBM50590486(CHEMBL5177168)
Affinity DataIC50: 0.514nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 155529BDBM155529(US9012461, 7 | US9012461, 5)
Affinity DataKd:  0.570nMpH: 7.4 T: 2°CAssay Description:Binding parameters of compounds were determined using a Biacore S51 sensor. An anti-GST antibody was immobilized onto a CM5 chip by primary amine-cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2015
Entry Details
US Patent

TargetFocal adhesion kinase 1(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50590473BDBM50590473(CHEMBL5192604)
Affinity DataIC50: 0.579nMAssay Description:Inhibition of recombinant human FAK (393 to 698 residues) using poly (4:1 Glu, Tyr) peptide as substrate incubated for 60 mins in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418649BDBM418649(N-methyl-4-{[4-({2- [methyl(methylsulfonyl)amino]b...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418650BDBM418650(N-ethyl-4-({4-[({3- [methyl(methylsulfonyl)amino]p...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418651BDBM418651(ethyl [4-({4-[({2- [methyl(methylsulfonyl)amino]py...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418609BDBM418609(N-methyl-4-({4-[({2- [methyl(methylsulfonyl)amino]...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418610BDBM418610(N-methyl-4-({4-[({6-methyl-2- [methyl(methylsulfon...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418604BDBM418604(3-methoxy-4-({4-[({2- [methyl(methylsuffonyl)amino...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418605BDBM418605(3-methoxy-4-({4-[({6-methyl-2- [methyl(methylsulfo...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418606BDBM418606(N-[3-({[2-anilino-5- (trifluoromethyl)pyrimidin-4-...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418607BDBM418607(N-[3-({[2-anilino-5- (trifluoromethyl)pyrimidin-4-...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418634BDBM418634(N-[5-({[2-anilino-5- (trifluoromethyl)pyrimidin-4-...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418603BDBM418603(3-methoxy-4-{[4-{[3- (methylsulfonyl)benzyl]amino}...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418597BDBM418597(methyl 4-({4-[({2- [methyl(methylsulfonyl)amino]py...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

TargetFocal adhesion kinase 1 [410-689](Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 418624BDBM418624(N-[2-(([2-anilino-5- (trifluoromethyl)pyrimidin-4-...)
Affinity DataIC50: 0.590nMAssay Description:The in vitro activity of the compounds of the compounds of the invention may be determined by the following procedure. More particularly, the followi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details
US Patent

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