Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]kianic acid from recombinant GluK2 kainate receptor (unknown origin) expressed in HEK293 cell membranes measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H](2S, 4R)-4-MeGlu (SYM-2081) from GluK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 18.3nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 29.8nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 31.7nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Compound was tested for agonistic activity at Glutamate receptor 6 using HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 38.4nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 41.1nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Compound was tested for binding affinity against human Ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]-kainate as radio...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]-kainate from human recombinant GluK2 receptor expressed in HEK293 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 54.3nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 57.4nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 82.2nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 90.6nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 93.5nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 129nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Displacement of [3H]-kainic acid from GluR6 (unknown origin) expressed in Sf9 cells membraneMore data for this Ligand-Target Pair
Affinity DataKi: 131nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 147nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 147nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 169nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 263nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 288nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 339nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Compound was tested for agonistic activity at Glutamate receptor 6 using HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 559nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 610nMAssay Description:Binding affinity for human GluR6 expressed in HEK293 cells using [3]H-kainateMore data for this Ligand-Target Pair
Affinity DataKi: 663nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 667nMAssay Description:Inhibition of [3H]kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Displacement of [3H]-kainate from GluK2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:Effective concentration against human GluR6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:Compound was tested for agonistic activity at Glutamate receptor 6 using HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 823nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 908nMAssay Description:Binding affinity to GluK2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity against human ionotropic glutamate receptor ionotropic kainate 2 in HEK293 cells using [3H]kainate as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.11E+3nMAssay Description:Binding affinity against human GluR6More data for this Ligand-Target Pair











3D Structure (crystal)































