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TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047418(CHEMBL3319223)
Affinity DataIC50: 3.40nMAssay Description:Displacement of [125I]human ghrelin from rat GHS-R1a expressed in HEK cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetHistone deacetylase 1/3/4/6/7(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047416(CHEMBL3319215)
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I]human ghrelin from rat GHS-R1a expressed in HEK cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50366958(CHEMBL1790587)
Affinity DataIC50: 6.30nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 5bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against histone deacetylase (HDAC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against rat liver histone deacetylase (HDAC) with substrate 3aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 13nMAssay Description:Inhibitory concentration against rat liver histone deacetylase (HDAC) with substrate 3bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50146077(CHEMBL3763388)
Affinity DataIC50: 18nMAssay Description:Inhibition of HDAC in rat liver by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against rat liver histone deacetylase (HDAC) with substrate 12aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50146076(CHEMBL3764525)
Affinity DataIC50: 21nMAssay Description:Inhibition of HDAC in rat liver by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50154337(6-((9S,13aR)-5-(S)-1-Benzyl-8,8-dimethyl-4,7,10,13...)
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 5bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration against rat liver histone deacetylase (HDAC) with substrate 5bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 26nMAssay Description:Inhibitory concentration against rat liver histone deacetylase (HDAC) with substrate 5aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475567(CHEMBL203207 | 6-Benzenesulfonylhexanoic Acid Hydr...)
Affinity DataIC50: 40nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50366958(CHEMBL1790587)
Affinity DataIC50: 56nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475570(CHEMBL201473 | 6-Benzenesulfinylhexanoic Acid Hydr...)
Affinity DataIC50: 60nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082325(CHEMBL99392)
Affinity DataIC50: 66nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 5bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082665(4-(dimethylamino)-N-(7-(hydroxyamino)-7-oxoheptyl)...)
Affinity DataIC50: 78nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50366958(CHEMBL1790587)
Affinity DataIC50: 80nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475559(CHEMBL371212)
Affinity DataIC50: 110nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475566(CHEMBL203028 | 6-Phenylsulfanylhexanoic Acid Hydro...)
Affinity DataIC50: 120nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50154337(6-((9S,13aR)-5-(S)-1-Benzyl-8,8-dimethyl-4,7,10,13...)
Affinity DataIC50: 137nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082665(4-(dimethylamino)-N-(7-(hydroxyamino)-7-oxoheptyl)...)
Affinity DataIC50: 148nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475565(CHEMBL198350 | 6-(4-Chlorophenylsulfinyl)Hexanoic ...)
Affinity DataIC50: 150nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082666(4-Dimethylamino-N-(5-hydroxycarbamoyl-pentyl)-benz...)
Affinity DataIC50: 152nMAssay Description:Inhibitory activity against histone deacetylase (HDAC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082666(4-Dimethylamino-N-(5-hydroxycarbamoyl-pentyl)-benz...)
Affinity DataIC50: 153nMAssay Description:Inhibitory concentration against rat liver histone deacetylase (HDAC) with substrate 3bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475562(CHEMBL383285)
Affinity DataIC50: 160nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475558(CHEMBL201710 | 6-(4-Dimethylaminophenylsulfinyl)He...)
Affinity DataIC50: 180nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082666(4-Dimethylamino-N-(5-hydroxycarbamoyl-pentyl)-benz...)
Affinity DataIC50: 216nMAssay Description:Inhibitory concentration against rat liver histone deacetylase (HDAC) with substrate 3aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50154337(6-((9S,13aR)-5-(S)-1-Benzyl-8,8-dimethyl-4,7,10,13...)
Affinity DataIC50: 226nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475557(CHEMBL203421)
Affinity DataIC50: 240nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082657(4-Dimethylamino-N-(7-hydroxycarbamoyl-heptyl)-benz...)
Affinity DataIC50: 241nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 5bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082657(4-Dimethylamino-N-(7-hydroxycarbamoyl-heptyl)-benz...)
Affinity DataIC50: 256nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475556(CHEMBL200980 | 6-(4-Chlorophenylsulfanyl)Hexanoic ...)
Affinity DataIC50: 260nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475563(CHEMBL199713)
Affinity DataIC50: 310nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475561(CHEMBL380339)
Affinity DataIC50: 340nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082325(CHEMBL99392)
Affinity DataIC50: 349nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50220740(CHEMBL55974)
Affinity DataIC50: 359nMAssay Description:Inhibitory activity against histone deacetylase (HDAC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2018
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475569(CHEMBL201131 | 7-(4-Chlorophenylsulfinyl)Heptanoic...)
Affinity DataIC50: 380nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475564(CHEMBL381561)
Affinity DataIC50: 390nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475560(CHEMBL203036)
Affinity DataIC50: 400nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475568(CHEMBL201075)
Affinity DataIC50: 410nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082325(CHEMBL99392)
Affinity DataIC50: 411nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 440nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082657(4-Dimethylamino-N-(7-hydroxycarbamoyl-heptyl)-benz...)
Affinity DataIC50: 488nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 3bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082666(4-Dimethylamino-N-(5-hydroxycarbamoyl-pentyl)-benz...)
Affinity DataIC50: 640nMAssay Description:Inhibitory concentration against rat liver histone deacetylase (HDAC) with substrate 5aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475571(CHEMBL199665)
Affinity DataIC50: 700nMAssay Description:Inhibition of HDAC in rat liver homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50146075(CHEMBL3765502)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of HDAC in rat liver by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50005711(GNF-Pf-1011 | CHEBI:46024 | TRICHOSTATIN | Trichos...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition concentration required to inhibit rat liver histone deacetylase (HDAC) in the presence of compound 5e as a substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50082665(4-(dimethylamino)-N-(7-(hydroxyamino)-7-oxoheptyl)...)
Affinity DataIC50: 3.51E+3nMAssay Description:Inhibitory activity against rat liver Histone deacetylase with substrate 5bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistone deacetylase(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50220741(CHEMBL417594)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibitory activity against histone deacetylase (HDAC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2018
Entry Details Article
PubMed
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