Compile Data Set for Download or QSAR
Report error Found 34 of affinity data for UniProtKB/TrEMBL: Q62194
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602486BDBM50602486(CHEMBL5196154)
Affinity DataKd:  13nMAssay Description:Binding affinity to MERTK in cuprizone-challenged C57BL/6 mouse whole brain assessed as dissociation constant at 18.1 nM by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50602486BDBM50602486(CHEMBL5196154)
Affinity DataKd:  20nMAssay Description:Binding affinity to MERTK in cuprizone-challenged C57BL/6 mouse brain CC/HC region assessed as dissociation constant at 18.1 nM by autoradiographyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571947BDBM50571947(CHEMBL4850929)
Affinity DataIC50: 24nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571953BDBM50571953(CHEMBL4860541)
Affinity DataIC50: 34nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571933BDBM50571933(CHEMBL4878216)
Affinity DataIC50: 34nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571932BDBM50571932(CHEMBL4865150)
Affinity DataIC50: 39nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571952BDBM50571952(CHEMBL4858396)
Affinity DataIC50: 51nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571944BDBM50571944(CHEMBL4856749)
Affinity DataIC50: 55nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571025BDBM50571025(CHEMBL4846932)
Affinity DataIC50: 61nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571943BDBM50571943(CHEMBL4848465)
Affinity DataIC50: 78nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571945BDBM50571945(CHEMBL4866147)
Affinity DataIC50: 79nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571935BDBM50571935(CHEMBL4878071)
Affinity DataIC50: 80nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571946BDBM50571946(CHEMBL4859513)
Affinity DataIC50: 92nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571931BDBM50571931(CHEMBL4875387)
Affinity DataIC50: 110nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571950BDBM50571950(CHEMBL4870464)
Affinity DataIC50: 110nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571949BDBM50571949(CHEMBL4874534)
Affinity DataIC50: 130nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571951BDBM50571951(CHEMBL4864780)
Affinity DataIC50: 130nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571940BDBM50571940(CHEMBL4859147)
Affinity DataIC50: 150nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571955BDBM50571955(CHEMBL4860402)
Affinity DataIC50: 180nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571954BDBM50571954(CHEMBL4857544)
Affinity DataIC50: 210nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571934BDBM50571934(CHEMBL4861291)
Affinity DataIC50: 240nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571925BDBM50571925(CHEMBL4852474)
Affinity DataIC50: 280nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571930BDBM50571930(CHEMBL4860139)
Affinity DataIC50: 280nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571939BDBM50571939(CHEMBL4858522)
Affinity DataIC50: 290nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571941BDBM50571941(CHEMBL4846790)
Affinity DataIC50: 370nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571942BDBM50571942(CHEMBL4851171)
Affinity DataIC50: 370nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571936BDBM50571936(CHEMBL4872556)
Affinity DataIC50: 440nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571927BDBM50571927(CHEMBL4870149)
Affinity DataIC50: 570nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571937BDBM50571937(CHEMBL4846861)
Affinity DataIC50: 630nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571929BDBM50571929(CHEMBL4860065)
Affinity DataIC50: 730nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571928BDBM50571928(CHEMBL4869791)
Affinity DataIC50: 810nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571938BDBM50571938(CHEMBL4875172)
Affinity DataIC50: 910nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571926BDBM50571926(CHEMBL4872079)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Monash University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50571948BDBM50571948(CHEMBL4870992)
Affinity DataIC50: 4.11E+3nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed