Compile Data Set for Download or QSAR
Report error Found 391 of affinity data for UniProtKB/TrEMBL: Q80SS6
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50156370(CHEMBL3793436)
Affinity DataEC50:  0.0620nMAssay Description:Agonist activity at mouse TGR5 expressed in CHO-K1 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2017
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50266580(CHEMBL4087611)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at mouse TGR5 transfected in HEK293 cells assessed as cAMP accumulation after overnight incubation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50266544(CHEMBL4060410)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at mouse TGR5 transfected in HEK293 cells assessed as cAMP accumulation after overnight incubation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM398287(US10323016, Example 26)
Affinity DataEC50:  0.5nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003570(CHEMBL3234869)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003559(CHEMBL3234570)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50614538(CHEMBL5286836)
Affinity DataEC50:  0.710nMAssay Description:Inhibition of mouse TGR5More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50266538(US10323016, Example 4 | CHEMBL4084668)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at mouse TGR5 transfected in HEK293 cells assessed as cAMP accumulation after overnight incubation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50266552(US10323016, Example 20 | CHEMBL4094487)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at mouse TGR5 transfected in HEK293 cells assessed as cAMP accumulation after overnight incubation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50019474(CHEMBL3290717)
Affinity DataEC50:  0.920nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells co-expressing CRE after 5.5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50399970(CHEMBL2181229)
Affinity DataEC50:  0.980nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells incubated for 5.5 hrs by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459101(CHEMBL4213913)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50266538(US10323016, Example 4 | CHEMBL4084668)
Affinity DataEC50:  1nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003573(CHEMBL3234871)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50266552(US10323016, Example 20 | CHEMBL4094487)
Affinity DataEC50:  1nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003407(CHEMBL3234568)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003569(CHEMBL3234868)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459099(CHEMBL4202981)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459099(CHEMBL4202981)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459141(CHEMBL4212707)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003567(CHEMBL3234582)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459138(CHEMBL4209799)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50399969(CHEMBL2181227)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells incubated for 5.5 hrs by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50266567(US10323016, Example 21 | CHEMBL4090147)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 transfected in HEK293 cells assessed as cAMP accumulation after overnight incubation by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459136(CHEMBL4204655)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459096(CHEMBL4217797)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003572(CHEMBL3234870)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459127(CHEMBL4209669)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003568(CHEMBL3234583)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003287(CHEMBL3234577)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50266567(US10323016, Example 21 | CHEMBL4090147)
Affinity DataEC50:  2nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2020
Entry Details
US Patent

TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50399968(CHEMBL2181228)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells incubated for 5.5 hrs by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621444(CHEMBL5394421)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621439(CHEMBL5437749)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621445(CHEMBL5422904)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621443(CHEMBL5415272)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50399967(CHEMBL2181230)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells incubated for 5.5 hrs by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621437(CHEMBL5427760)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621438(CHEMBL5414305)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50019475(CHEMBL3290716)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells co-expressing CRE after 5.5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621440(CHEMBL5395284)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459140(CHEMBL4218746)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459145(CHEMBL4207707)
Affinity DataEC50:  2.5nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621442(CHEMBL5439914)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003336(CHEMBL3234565)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50003561(CHEMBL3234571)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50399962(CHEMBL2181239)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at mouse TGR5 transfected in HEK293T cells assessed intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50459124(CHEMBL4209927)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at mouse TGR5 expressed in HEK293 cells assessed as increase in intracellular cAMP level by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621446(CHEMBL5398966)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50621441(CHEMBL5413666)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at mouse TGR5 expressed in human HEK293 cells co-expressing CRE-driven luciferase reporter gene assessed as luciferase activity incu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
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