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TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM11695((2S)-1-{2-[(3-hydroxyadamantan-1-yl)amino]acetyl}p...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of human recombinant DPP9 using Gly-Pro-AMC as substrate preincubated for 15 mins followed by substrate addition and measured for 20 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324512(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methyl-N-...)
Affinity DataKi:  0.190nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324510(1-(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methyl...)
Affinity DataKi:  0.280nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442192(CHEMBL2441845)
Affinity DataKi:  0.300nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324511(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methyl-N-...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50389480(CHEMBL2063040)
Affinity DataIC50: 0.310nMAssay Description:Inhibition of human DPP9 expressed in HEK293 cells using Ala-Pro-p-nitroanilide hydrochloride salt as substrate preincubated for 10 mins prior to add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50050511((R)-1-(2-aminoacetyl)pyrrolidin-2-ylboronic acid |...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442198(CHEMBL2441839)
Affinity DataKi:  0.5nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataKi:  0.530nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324504(6-(aminomethyl)-5-(2,4-dichlorophenyl)-N,7-dimethy...)
Affinity DataKi:  0.550nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324500(1-(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methyl...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataKi:  0.760nMAssay Description:Inhibition of human recombinant DPP9 expressed in HEK293T cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442183(CHEMBL2441955)
Affinity DataKi:  0.800nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324524((6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylim...)
Affinity DataKi:  0.830nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324505(6-(aminomethyl)-5-(2,4-dichlorophenyl)-N,7-dimethy...)
Affinity DataKi:  0.860nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324494(6-(aminomethyl)-5-(2,4-dichlorophenyl)-N-(1,3-dime...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442193(CHEMBL2441844)
Affinity DataKi:  0.900nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324501(6-(aminomethyl)-5-(2,4-dichlorophenyl)-N-(1-ethyl-...)
Affinity DataKi:  0.900nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442184(CHEMBL2441954)
Affinity DataKi:  0.900nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324497((6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylim...)
Affinity DataKi:  0.940nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50629038(CHEMBL5425473)
Affinity DataIC50: 1nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324516((6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylim...)
Affinity DataKi:  1nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM142093(US8933056, Chg-boroPro Thioxamide | US8933056, Chg...)
Affinity DataIC50: 1.10nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442206(CHEMBL2441831)
Affinity DataKi:  1.20nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442191(CHEMBL2441846)
Affinity DataKi:  1.30nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442181(CHEMBL2441829)
Affinity DataKi:  1.30nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324522((6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylim...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324515(6-(aminomethyl)-5-(2,4-dichlorophenyl)-N,N-diethyl...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324518(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methyl-N-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM514555(US11096924, DASH-inhibitors 4367 | US11583516, Cmp...)
Affinity DataIC50: 1.5nMAssay Description:Materials: Enzymes Recombinant human DPPIV (R&D Systems, Cat. No. 1180-SE). Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527). Recombin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM514555(US11096924, DASH-inhibitors 4367 | US11583516, Cmp...)
Affinity DataIC50: 1.5nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50050516(Boronic acid derivative | CHEMBL63726 | US11096924...)
Affinity DataIC50: 1.60nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50612314(CHEMBL5279548)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of DPP-9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 1.70nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442185(CHEMBL2441953)
Affinity DataKi:  1.80nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50050520(Boronic acid derivative | CHEMBL63406 | US11096924...)
Affinity DataIC50: 1.90nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324521(4-(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methyl...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442201(CHEMBL2441836)
Affinity DataKi:  1.90nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442201(CHEMBL2441836)
Affinity DataKi:  1.90nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324508(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methyl-N-...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324525(6-(aminomethyl)-5-(2,4-dichlorophenyl)-N,7-dimethy...)
Affinity DataKi:  2nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50369128(CHEMBL1790483 | US11096924, DASH-inhibitors 4316 |...)
Affinity DataIC50: 2nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
US Patent

TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50171552((S)-2-(S)-Amino-1-(2-boron-dihydroxide-pyrrolidine...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against human dipeptidylpeptidase 9 using FP-TAMRA incubated for 30 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50389473(CHEMBL2063033)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human DPP9 expressed in HEK293 cells using Ala-Pro-p-nitroanilide hydrochloride salt as substrate preincubated for 10 mins prior to add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324513(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methyl-N-...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324523(N-((3S)-1-(6-(aminomethyl)-5-(2,4-dichlorophenyl)-...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human DPP9 using H-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50324517((6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylim...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of human DPP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Sichuan Normal University

Curated by ChEMBL
LigandPNGBDBM50442180(CHEMBL2441830)
Affinity DataKi:  2.30nMAssay Description:Inhibition of DPP9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
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