Compile Data Set for Download or QSAR
Report error Found 30 of affinity data for UniProtKB/TrEMBL: Q8I6Z5
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50514481BDBM50514481(CHEMBL3782104)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant Plasmodium falciparum Plasmepsin 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50500851BDBM50500851(CHEMBL3780033)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of Plasmodium falciparum PMV assessed as fluorogenic substrate cleavage using DABCYL-RNKRTLAQKQ-E-EDANS as fluorogenic substrate after 120...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/4/2020
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099406BDBM50099406(CHEMBL3344272)
Affinity DataIC50: 19nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099378BDBM50099378(CHEMBL3344165)
Affinity DataIC50: 26nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099272BDBM50099272(CHEMBL3344164)
Affinity DataIC50: 29nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099380BDBM50099380(CHEMBL3344166)
Affinity DataIC50: 77nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099381BDBM50099381(CHEMBL3344261)
Affinity DataIC50: 230nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099391BDBM50099391(CHEMBL3344266)
Affinity DataIC50: 348nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099395BDBM50099395(CHEMBL3344270)
Affinity DataIC50: 378nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099387BDBM50099387(CHEMBL3344262)
Affinity DataIC50: 530nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099394BDBM50099394(CHEMBL3344269)
Affinity DataIC50: 550nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099148BDBM50099148(CHEMBL3344151)
Affinity DataIC50: 556nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099390BDBM50099390(CHEMBL3344265)
Affinity DataIC50: 569nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099171BDBM50099171(CHEMBL3344152)
Affinity DataIC50: 613nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099240BDBM50099240(CHEMBL3344157)
Affinity DataIC50: 614nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099388BDBM50099388(CHEMBL3344263)
Affinity DataIC50: 622nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099403BDBM50099403(CHEMBL3344271)
Affinity DataIC50: 625nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099389BDBM50099389(CHEMBL3344264)
Affinity DataIC50: 772nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099393BDBM50099393(CHEMBL3344268)
Affinity DataIC50: 774nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099236BDBM50099236(CHEMBL3344153)
Affinity DataIC50: 865nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099237BDBM50099237(CHEMBL3344154)
Affinity DataIC50: 967nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099392BDBM50099392(CHEMBL3344267)
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099241BDBM50099241(CHEMBL3344158)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099242BDBM50099242(CHEMBL3344159)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099243BDBM50099243(CHEMBL3344160)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099247BDBM50099247(CHEMBL3344161)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099249BDBM50099249(CHEMBL3344162)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099252BDBM50099252(CHEMBL3344163)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099238BDBM50099238(CHEMBL3344155)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed
TargetPlasmepsin V(Plasmodium falciparum (isolate 3D7))
University of Zambia

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099239BDBM50099239(CHEMBL3344156)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Plasmodium falciparum plasmepsin V assessed as cleavage of wtKAHRP fluorogenic substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2016
Entry Details Article
PubMed