Compile Data Set for Download or QSAR
Report error Found 160 of affinity data for UniProtKB/TrEMBL: Q9UK84
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118219BDBM50118219(Bz-ATP | CHEMBL339386)
Affinity DataEC50:  2nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 526264BDBM526264(US11185100, TABLE 14.4)
Affinity DataIC50: 3.5nMAssay Description:Agonist activity at human P2X1R expressing CHO cells assessed as reduction in intracellular Ca2+ influx pretreated with Fluo-4 for 1 hr followed by c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370141BDBM50370141(TNP-ATP)
Affinity DataEC50:  6nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430160BDBM50430160(TCMDC-125465 | CHEMBL536151)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430195BDBM50430195(CHEMBL2338696)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430185BDBM50430185(CHEMBL2179173)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540434BDBM50540434(CHEMBL4640175)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430177BDBM50430177(CHEMBL2088014)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540436BDBM50540436(CHEMBL2179174)
Affinity DataIC50: 51nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118232BDBM50118232(ATP, 2-meS | CHEMBL336208 | 2-MeSATP)
Affinity DataEC50:  54nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366480BDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  56nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430156BDBM50430156(CHEMBL2338695)
Affinity DataIC50: 58nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50422739BDBM50422739(CHEMBL413145)
Affinity DataIC50: 63nMAssay Description:Inhibitory concentration against human P2X purinoceptor 1 expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540422BDBM50540422(CHEMBL4644398)
Affinity DataIC50: 71nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540442BDBM50540442(CHEMBL2088011)
Affinity DataIC50: 76nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430159BDBM50430159(CHEMBL461542)
Affinity DataIC50: 77nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430176BDBM50430176(MMV665807 | SJ000010289 | CHEMBL589733)
Affinity DataIC50: 91nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540410BDBM50540410(CHEMBL337395)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human P2X1R transfected in CHO-K1 cells preincubated for 30 mins followed by alpha,beta-meATP addition by luminescence based a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540439BDBM50540439(CHEMBL2088009)
Affinity DataIC50: 172nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015276BDBM50015276(CHEMBL3263056 | US9428504, 166 | US9428504, 167)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at P2X1 receptor (unknown origin) by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2015
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118220BDBM50118220(adenosine(5')tetraphospho(5')adenosine | P(1),P(4)...)
Affinity DataEC50:  182nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540432BDBM50540432(CHEMBL2088012)
Affinity DataIC50: 199nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118221BDBM50118221(alpha,beta-meATP | DIPHOSPHOMETHYLPHOSPHONIC ACID ...)
Affinity DataEC50:  200nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118228BDBM50118228(5,7-Disulfo-4-(3-{3-[3-(4,6,8-trisulfo-naphthalen-...)
Affinity DataIC50: 210nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540449BDBM50540449(CHEMBL4637528)
Affinity DataIC50: 219nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430194BDBM50430194(CHEMBL2313115)
Affinity DataIC50: 236nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240455BDBM50240455(CHEMBL1253351)
Affinity DataIC50: 236nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430186BDBM50430186(CHEMBL2178702)
Affinity DataIC50: 323nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540443BDBM50540443(CHEMBL4648128)
Affinity DataIC50: 335nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430170BDBM50430170(CHEMBL2338686)
Affinity DataIC50: 341nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540456BDBM50540456(CHEMBL2313133)
Affinity DataIC50: 439nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50168286BDBM50168286(1H-Benzoimidazole-2-carboxylic acid [(R)-1-((1S,2R...)
Affinity DataIC50: 496nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540441BDBM50540441(CHEMBL2179168)
Affinity DataIC50: 522nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540444BDBM50540444(CHEMBL2179170)
Affinity DataIC50: 567nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430160BDBM50430160(TCMDC-125465 | CHEMBL536151)
Affinity DataIC50: 570nMAssay Description:Antagonist activity P2X1 receptor in Apyrase pre-treated human platelets assessed as inhibition of collagen-induced platelet aggregation pre-incubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50399190BDBM50399190(CHEMBL2180149)
Affinity DataIC50: 602nMAssay Description:Antagonist activity at human P2X1 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540423BDBM50540423(CHEMBL4639803)
Affinity DataIC50: 655nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430193BDBM50430193(CHEMBL2313119)
Affinity DataIC50: 755nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540424BDBM50540424(CHEMBL3628655)
Affinity DataIC50: 869nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540433BDBM50540433(CHEMBL2312822)
Affinity DataIC50: 907nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540435BDBM50540435(CHEMBL4634436)
Affinity DataIC50: 915nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540413BDBM50540413(CHEMBL2313124)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 85682BDBM85682(CAS_5311315 | NSC_5311315 | NF279)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50171290BDBM50171290(SR 147778 | CHEMBL189676 | 5-(4-Bromo-phenyl)-1-(2...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50430195BDBM50430195(CHEMBL2338696)
Affinity DataIC50: 1.14E+3nMAssay Description:Antagonist activity P2X1 receptor in Apyrase pre-treated human platelets assessed as inhibition of collagen-induced platelet aggregation pre-incubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118229BDBM50118229(MRS 2179 | CHEMBL129841)
Affinity DataEC50:  1.15E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 )More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118229BDBM50118229(MRS 2179 | CHEMBL129841)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of P2X1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118229BDBM50118229(MRS 2179 | CHEMBL129841)
Affinity DataIC50: 1.15E+3nMAssay Description:Affinity at P2X purinoceptor 1 (P2X1) and the value is expressed as IC50More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540430BDBM50540430(Salfluverine)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 1(Human)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50540445BDBM50540445(CHEMBL2179166)
Affinity DataIC50: 1.34E+3nMAssay Description:Antagonist activity at non-desensitizing human P2X1 receptor ( P2X2/P2X1 chimera) expressed in human 1321N1 cells assessed as inhibition of ATP-induc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
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