Compile Data Set for Download or QSAR
Report error Found 372 of affinity data for UniProtKB/TrEMBL: Q9ULU5
TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572231BDBM572231(US11447505, Example E236 | 3-[4-[(6S)-1,8-diazaspi...)
Affinity DataKi:  0.0120nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572232BDBM572232(3-[4-[(6S)-1,8-diazaspiro[5.5]undecan-8-yl]-1H- py...)
Affinity DataKi:  0.0150nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572233BDBM572233(US11447505, Example E168 | (6S)-8-(3-pyrimidin-4-y...)
Affinity DataKi:  0.0230nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572234BDBM572234(2-[4-[(6S)-1,8-diazaspiro[5.5]undecan-8-yl]-1H- py...)
Affinity DataKi:  0.0250nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572235BDBM572235((6S)-8-(3-pyridazin-4-yl-1H-pyrrolo[2,3-b]pyridin-...)
Affinity DataKi:  0.0260nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572236BDBM572236((6S)-1-methyl-8-(3-pyrimidin-4-yl-1H-pyrrolo[2,3- ...)
Affinity DataKi:  0.0280nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572237BDBM572237(2-[4-[(5S)-2,6-diazaspiro[4.5]decan-2-yl]-1H- pyrr...)
Affinity DataKi:  0.0300nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572239BDBM572239((6S)-8-[3-(2-pyridyl)-1H-pyrrolo[2,3-b]pyridin-4-y...)
Affinity DataKi:  0.0390nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572238BDBM572238(2-[4-(1-ethyl-1,8-diazaspiro[5.5]undecan-8-yl)-1H-...)
Affinity DataKi:  0.0390nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572240BDBM572240((6S)-1-ethyl-8-(3-pyrimidin-4-yl-1H-pyrrolo[2,3- b...)
Affinity DataKi:  0.0400nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572241BDBM572241(3-[4-(1,8- diazaspiro[5.5]undecan- 8-yl)-1H-pyrrol...)
Affinity DataKi:  0.0490nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572242BDBM572242(2-[4-[(6S)-1,8-diazaspiro[5.5]undecan-8-yl]-1H- py...)
Affinity DataKi:  0.0540nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572243BDBM572243((5S)-2-(3-pyrimidin-5-yl-1H-pyrrolo[2,3-b]pyridin-...)
Affinity DataKi:  0.0570nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572244BDBM572244(2-[4-[(5S)-2,6-diazaspiro[4.5]decan-2-yl]-1H- pyrr...)
Affinity DataKi:  0.0600nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572245BDBM572245(2-[4-(1,8- diazaspiro[5.5]undecan-8- yl)-1H-pyrrol...)
Affinity DataKi:  0.0630nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572246BDBM572246(2-[4-(1-ethyl-1,8-diazaspiro[5.5]undecan-8-yl)-1H-...)
Affinity DataKi:  0.0630nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572233BDBM572233(US11447505, Example E168 | (6S)-8-(3-pyrimidin-4-y...)
Affinity DataKi:  0.0650nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572249BDBM572249((5S)-2-(3-pyrimidin-4-yl-1H-pyrrolo[2,3-b]pyridin-...)
Affinity DataKi:  0.0650nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572247BDBM572247(8-[3-(5-fluoro-3-pyridyl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  0.0650nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572250BDBM572250(8-[3-(2-pyridyl)-1H- pyrrolo[2,3-b]pyridin-4- yl]-...)
Affinity DataKi:  0.0730nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572251BDBM572251(4-[4-(1,8-diazaspiro[5.5]undecan-8-yl)-1H-pyrrolo[...)
Affinity DataKi:  0.0810nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572252BDBM572252(2-[4-(2,6-diazaspiro[4.5]decan-2-yl)-1H-pyrrolo[2,...)
Affinity DataKi:  0.0820nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572253BDBM572253(3-ethyl-1-[3-(5-methylthiazol-2-yl)-1H-pyrrolo[2,3...)
Affinity DataKi:  0.0890nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572231BDBM572231(US11447505, Example E236 | 3-[4-[(6S)-1,8-diazaspi...)
Affinity DataKi:  0.0900nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572256BDBM572256(2-[4-(1,8- diazaspiro[5.5]undecan-8- yl)-1H-pyrrol...)
Affinity DataKi:  0.0920nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572255BDBM572255(3-methyl-1-(3-thiazol-2-yl-1H-pyrrolo[2,3-b]pyridi...)
Affinity DataKi:  0.0920nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572257BDBM572257(8-[3-(5-fluoro-2-pyridyl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  0.100nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572258BDBM572258(8-[3-(3-fluoro-2-pyridyl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  0.106nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572259BDBM572259(3-[4-(1,7-diazaspiro[4.4]nonan-7-yl)-1H-pyrrolo[2,...)
Affinity DataKi:  0.120nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572260BDBM572260(3-pyrimidin-4-yl-4- [[(3R)-3-piperidyl[oxy]- 1H-py...)
Affinity DataKi:  0.144nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572261BDBM572261(2-[4-(2,6- diazaspiro[4.5]decan-2- yl)-1H-pyrrolo[...)
Affinity DataKi:  0.154nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572262BDBM572262((3S)-N-methyl-1-(3-pyrimidin-4-yl-1H-pyrrolo[2,3- ...)
Affinity DataKi:  0.170nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572263BDBM572263(4-[(6S)-1,8-diazaspiro[5.5]undecan-8-yl]-1H- pyrro...)
Affinity DataKi:  0.179nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572264BDBM572264(3-methyl-1-(3-pyrimidin-5-yl-1H-pyrrolo[2,3-b]pyri...)
Affinity DataKi:  0.181nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572265BDBM572265(US11447505, Example E212)
Affinity DataKi:  0.184nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572266BDBM572266(US11447505, Example E41)
Affinity DataKi:  0.202nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572267BDBM572267(3-[4-(1,8-diazaspiro[5.5]undecan-8-yl)-1H-pyrrolo[...)
Affinity DataKi:  0.203nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572268BDBM572268(3-[4-(2,6-diazaspiro[4.5]decan-2-yl)-1H-pyrrolo[2,...)
Affinity DataKi:  0.206nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572269BDBM572269(2-(3-pyridazin-4-yl-1H- pyrrolo[2,3-b]pyridin-4-yl...)
Affinity DataKi:  0.219nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572270BDBM572270((3S)-N-cyclopropyl-1-(3-pyridazin-4-yl-1H-pyrrolo[...)
Affinity DataKi:  0.238nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572271BDBM572271(4-(1,8- diazaspiro[5.5]undecan-8- yl)-1H-pyrrolo[2...)
Affinity DataKi:  0.249nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572272BDBM572272((3S)-1-(3-isothiazol-4-yl- 1H-pyrrolo[2,3-b]pyridi...)
Affinity DataKi:  0.273nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572273BDBM572273(2-[4-[(5S)-1,7-diazaspiro[4.4]nonan-7-yl]-1H- pyrr...)
Affinity DataKi:  0.303nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572274BDBM572274((3S)-N-methyl-1-(3-thiazol-2-yl-1H-pyrrolo[2,3- b]...)
Affinity DataKi:  0.304nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572275BDBM572275(4-fluoro-1-(3-pyrimidin-4- yl-1H-pyrrolo[2,3- b]py...)
Affinity DataKi:  0.323nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572276BDBM572276(4-(1-ethyl-1,8-diazaspiro[5.5]undecan-8-yl)-1H- py...)
Affinity DataKi:  0.351nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572277BDBM572277(2-[4-(1,8- diazaspiro[5.5]undecan-8- yl)-1H-pyrrol...)
Affinity DataKi:  0.360nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572278BDBM572278(2-[4-(1,7- diazaspiro[4.4]nonan-7- yl)-1H-pyrrolo[...)
Affinity DataKi:  0.370nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572280BDBM572280((3S)-N-methyl-1-[3-(2- pyridyl)-1H-pyrrolo[2,3- b]...)
Affinity DataKi:  0.506nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

TargetSerine/threonine-protein kinase MRCK beta(Human)
Cancer Research Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 572281BDBM572281(2-[3-(2-pyridyl)-1H- pyrrolo[2,3-b]pyridin-4- yl]-...)
Affinity DataKi:  0.549nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2022
Entry Details
US Patent

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