Compile Data Set for Download or QSAR
Report error Found 85 for UniProtKB: Q9W535
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50326777BDBM50326777((2beta,3beta,5beta,22R)-2,3,14,20,22,25-hexahydrox...)
Affinity DataIC50: 46nMAssay Description:Binding affinity to Drosophila melanogaster EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488497BDBM50488497(CHEMBL2286719)
Affinity DataEC50:  219nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488514BDBM50488514(CHEMBL2286720)
Affinity DataEC50:  219nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataKi:  251nMAssay Description:Binding affinity to Drosophila melanogaster EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataEC50:  525nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488500BDBM50488500(CHEMBL2286737)
Affinity DataEC50:  794nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488484BDBM50488484(CHEMBL2286739)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178990BDBM50178990(CHEMBL2286425)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488517BDBM50488517(CHEMBL2286738)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488468BDBM50488468(CHEMBL2286448)
Affinity DataEC50: <1.32E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50226672BDBM50226672(makisterone A | CHEMBL255034)
Affinity DataIC50: 1.38E+3nMAssay Description:Binding affinity to Drosophila melanogaster EcRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488467BDBM50488467(CHEBI:38457 | RH-5849)
Affinity DataEC50:  1.82E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488516BDBM50488516(CHEMBL2286743)
Affinity DataEC50:  2.57E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488473BDBM50488473(CHEMBL2286426)
Affinity DataEC50:  2.82E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488497BDBM50488497(CHEMBL2286719)
Affinity DataEC50:  3.24E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488443BDBM50488443(CHEMBL2286420)
Affinity DataEC50:  3.63E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488499BDBM50488499(CHEMBL2228437)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488515BDBM50488515(CHEMBL2286740)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488456BDBM50488456(CHEMBL2286431)
Affinity DataEC50:  5.50E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488494BDBM50488494(CHEMBL2286736)
Affinity DataEC50:  6.17E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster B2 cells assessed as reduction in cell densityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178988BDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataEC50:  6.61E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488473BDBM50488473(CHEMBL2286426)
Affinity DataEC50:  6.92E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster Kc cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488508BDBM50488508(CHEMBL2286946)
Affinity DataEC50:  7.08E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor/Protein ultraspiracle(Fruit fly)
Ghent University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488482BDBM50488482(CHEMBL2286721)
Affinity DataEC50:  7.76E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488461BDBM50488461(CHEBI:38451 | Halofenozide)
Affinity DataEC50:  7.76E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488479BDBM50488479(CHEMBL2228435)
Affinity DataEC50:  8.51E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488458BDBM50488458(CHEMBL2286427)
Affinity DataEC50:  9.77E+3nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488477BDBM50488477(CHEMBL2286417)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50128314BDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488437BDBM50488437(CHEMBL2286416)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488495BDBM50488495(CHEMBL2286703)
Affinity DataEC50:  1.05E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488528BDBM50488528(CHEMBL2286728)
Affinity DataEC50:  1.12E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488476BDBM50488476(CHEMBL2286429)
Affinity DataEC50:  1.12E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488496BDBM50488496(CHEMBL2286722)
Affinity DataEC50:  1.15E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488490BDBM50488490(CHEMBL2286729)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488441BDBM50488441(CHEMBL2286428)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488489BDBM50488489(CHEMBL2286747)
Affinity DataEC50:  1.32E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488514BDBM50488514(CHEMBL2286720)
Affinity DataEC50:  1.55E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488484BDBM50488484(CHEMBL2286739)
Affinity DataEC50:  1.55E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488481BDBM50488481(CHEMBL2228859)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488507BDBM50488507(CHEMBL2286723)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50128305BDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50178990BDBM50178990(CHEMBL2286425)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488474BDBM50488474(CHEMBL2286423)
Affinity DataEC50:  2.57E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488533BDBM50488533(CHEMBL2286746)
Affinity DataEC50:  2.57E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488443BDBM50488443(CHEMBL2286420)
Affinity DataEC50:  3.39E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488475BDBM50488475(CHEMBL2286422)
Affinity DataEC50:  3.39E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488487BDBM50488487(CHEMBL2286748)
Affinity DataEC50:  3.63E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488467BDBM50488467(CHEBI:38457 | RH-5849)
Affinity DataEC50:  3.72E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetProtein ultraspiracle(Fruit fly)
Csiro Materials Science and Engineering and Csiro Food and Nutritional Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50488531BDBM50488531(CHEMBL2286751)
Affinity DataEC50:  3.72E+4nMAssay Description:Agonist activity at ecdysone receptor in Drosophila melanogaster S2 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
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