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Found 137 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily KQT member 1'
TargetPotassium voltage-gated channel subfamily KQT member 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)
Affinity DataKi:  1.06E+3nMAssay Description:Binding affinity at Voltage-gated potassium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279436(1-(2,3-dihydro-6-methoxychromen-4-ylideneamino)-3-...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106179(CHEMBL125327 | Enantiomer-4-(3-Butyl-[1,2,4]oxadia...)
Affinity DataIC50:  2nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279740(1-(2,3-dihydro-6-propoxychromen-4-ylideneamino)-3-...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279471(1-(2,3-dihydro-6-chlorochromen-4-ylideneamino)-3-(...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106169(CHEMBL338973 | Enantiomer-4-(3-Butyl-[1,2,4]oxadia...)
Affinity DataIC50:  9nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279454(1-(2,3-dihydro-6-propoxychromen-4-ylideneamino)-3-...)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106167(CHEMBL125000 | Enantiomer-4-(3-Cyclopropylmethyl-[...)
Affinity DataIC50:  18nMAssay Description:Bindind affinity value obtained by measuring the displacement of radioligand [3H]-(-)-cytisine from whole rat brain Nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106167(CHEMBL125000 | Enantiomer-4-(3-Cyclopropylmethyl-[...)
Affinity DataIC50:  18nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279703(1-(6-butoxy-2,3-dihydrochromen-4-ylideneamino)-3-(...)
Affinity DataIC50:  22nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106178(4-(3-Butyl-[1,2,4]oxadiazol-5-yl)-N-(3,3-dimethyl-...)
Affinity DataIC50:  23nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106168(CHEMBL124448 | Enantiomer-N-(2,2-Dimethyl-cyclopen...)
Affinity DataIC50:  27nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279453(1-(6-ethoxy-2,3-dihydrochromen-4-ylideneamino)-3-(...)
Affinity DataIC50:  27nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106168(CHEMBL124448 | Enantiomer-N-(2,2-Dimethyl-cyclopen...)
Affinity DataIC50:  27nMAssay Description:Bindind affinity value obtained by measuring the displacement of radioligand [3H]-(-)-cytisine from whole rat brain Nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50061218((E)-3-(2,4-Dichloro-phenyl)-N-((R)-1-methyl-2-oxo-...)
Affinity DataIC50:  31nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106176(CHEMBL340681 | Enantiomer-N-(2,2-Dimethyl-cyclopen...)
Affinity DataIC50:  40nMAssay Description:Bindind affinity values obtained by measuring the displacement of radioligand [3H]-(-)-cytisine from a preparation of whole rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106176(CHEMBL340681 | Enantiomer-N-(2,2-Dimethyl-cyclopen...)
Affinity DataIC50:  40nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279717(1-(2,3-dihydro-6-chlorochromen-4-ylideneamino)-3-(...)
Affinity DataIC50:  73nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50099582((3R,4S)N-[3-Hydroxy-2,2-dimethyl-6-(4,4,4-trifluor...)
Affinity DataIC50:  120nMAssay Description:Inhibition of guinea pig Iks potassium channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106182(CHEMBL123085 | N-(3,3-Dimethyl-butyl)-4-(3-phenyl-...)
Affinity DataIC50:  130nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50117913((E)-1-((5-(4-chlorophenyl)furan-2-yl)methyleneamin...)
Affinity DataIC50:  240nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106166(CHEMBL122341 | N-(3,3-Dimethyl-butyl)-4-hexyloxy-b...)
Affinity DataIC50:  250nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106177(CHEMBL431682 | N-(3,3-Dimethyl-butyl)-4-indol-1-yl...)
Affinity DataIC50:  260nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279456(1-(2,3-dihydro-6-methylchromen-4-ylideneamino)-3-(...)
Affinity DataIC50:  304nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279719(1-(2,3-dihydro-6-amidecarboxylchromen-4-ylideneami...)
Affinity DataIC50:  330nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106184(CHEMBL121751 | N-(3,3-Dimethyl-cyclopentyl)-4-hexy...)
Affinity DataIC50:  360nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106180(CHEMBL124595 | N-(3,3-Dimethyl-cyclohexylmethyl)-4...)
Affinity DataIC50:  370nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106181(Biphenyl-4-carboxylic acid (3,3-dimethyl-butyl)-am...)
Affinity DataIC50:  540nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106164(CHEMBL123569 | Enantiomer-N-(2,2-Dimethyl-cyclopen...)
Affinity DataIC50:  580nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106164(CHEMBL123569 | Enantiomer-N-(2,2-Dimethyl-cyclopen...)
Affinity DataIC50:  580nMAssay Description:Bindind affinity value obtained by measuring the displacement of radioligand [3H]-(-)-cytisine from a preparation of whole rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279700(1-(2,3-dihydro-6-methoxychromen-4-ylideneamino)-3-...)
Affinity DataIC50:  650nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106175(CHEMBL121750 | Enantiomer-N-(2,2-Dimethyl-cyclopen...)
Affinity DataIC50:  710nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106175(CHEMBL121750 | Enantiomer-N-(2,2-Dimethyl-cyclopen...)
Affinity DataIC50:  710nMAssay Description:Bindind affinity value obtained by measuring the displacement of radioligand [3H]-(-)-cytisine from whole rat brain Nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50371391(SENICAPOC)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of voltage-gated K channel 7.1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279741(1-(6-butoxy-2,3-dihydrochromen-4-ylideneamino)-3-(...)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279739(1-(6-ethoxy-2,3-dihydrochromen-4-ylideneamino)-3-(...)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279455(1-(6-butoxy-2,3-dihydrochromen-4-ylideneamino)-3-(...)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50279702(1-(2,3-dihydro-6-propoxychromen-4-ylideneamino)-3-...)
Affinity DataIC50:  1.28E+3nMAssay Description:Inhibition of KVLQT1/minK in guinea pig ventricular myocytes assessed as blockade of slow delayed rectifier potassium current by whole cell patch-cla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106174(CHEMBL332297 | N-(2,2-Dimethyl-cyclohexylmethyl)-4...)
Affinity DataIC50:  1.40E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50254401(CHEMBL4093377)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of KCNQ1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50254387(CHEMBL4062193)
Affinity DataIC50:  2.64E+3nMAssay Description:Inhibition of KCNQ1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50395464(CHEMBL2164048)
Affinity DataIC50:  2.92E+3nMAssay Description:Antagonist activity at KCNQ1 expressed in CHO cells incubated for 3 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50254388(CHEMBL4101680)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of KCNQ1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106174(CHEMBL332297 | N-(2,2-Dimethyl-cyclohexylmethyl)-4...)
Affinity DataIC50: >3.00E+3nMAssay Description:Bindind affinity value obtained by measuring the displacement of radioligand [3H]-(-)-cytisine from a preparation of whole rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106165((3-tert-Butyl-pyrrolidin-1-yl)-(4-hexyloxy-phenyl)...)
Affinity DataIC50: >3.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106170(CHEMBL122865 | N-(2-Diethylamino-ethyl)-4-hexyloxy...)
Affinity DataIC50:  3.50E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106183(1-(4-(Hexyloxy)phenyl)-3-(piperidin-1-yl)propan-1-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106171(CHEMBL122637 | Diethyl-{2-[4-(1,1,3,3-tetramethyl-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106173(CHEMBL341368 | N,N-Diethyl-2-[4-(1,1,3,3-tetrameth...)
Affinity DataIC50:  5.00E+3nMAssay Description:Molar concentration required to inhibit 50% of the activating delayed-rectifier K+ current in isolated guinea pig ventricularmyocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 1(Cavia porcellus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50106227((3R,4S)-Ethanesulfonic acid (6-cyano-3-hydroxy-2,2...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of guinea pig Iks potassium channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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