Affinity DataIC50: 130nMAssay Description:Inhibition of Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 600nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri ES114 LuxR after 4 to 8 hrs by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR transfected with lasB-GFP by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Antagonist activity at LasR in Pseudomonas aeruginosa harboring plasI-LVAgfp assessed as inhibition of GFP production incubated for 6 hrs by fluoresc...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+4nMAssay Description:Antagonist activity at Aliivibrio fischeri LuxR by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR transfected with lasB-GFP by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR transfected with lasB-GFP by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at Pseudomonas aeruginosa LasR transfected with lasB-GFP by luminescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair
TargetTranscriptional activator protein LasR(Pseudomonas aeruginosa)
Larkin University
Curated by ChEMBL
Larkin University
Curated by ChEMBL
Affinity DataIC50: 1.16E+5nMAssay Description:Inhibition of LasR in Pseudomonas aeruginosa PAO-JP2 harboring plasI-LVAgfp incubated for 6 hrs by fluorescence methodMore data for this Ligand-Target Pair