Affinity DataIC50: 8.79E+3nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Compound was evaluated for the agonistic activity towards 5-hydroxytryptamine 4 receptor using the rat tunica muscularis mucosae (TMM) esophagus stri...More data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: >2.00E+4nMAssay Description:Activity at human beta1 adrenergic receptorMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: 2.99E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Dissociation constant against EPSP synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Nav1.5 by electrophysiology methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: 3.94E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck
Curated by ChEMBL
Merck
Curated by ChEMBL
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 65nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
Affinity DataEC50: 26nMAssay Description:Inhibition of NET (unknown origin) expressed in HEK293 cells assessed as reduction in norepinephrine reuptakeMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Agonist activity at human beta3 adrenergic receptorMore data for this Ligand-Target Pair