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Found 68 with Last Name = 'afzal' and Initial = 'o'
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50065646(CHEMBL3087181)
Affinity DataIC50: <0.400nMAssay Description:Inhibition of human MAGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50242634(5-((biphenyl-4-yl)methyl)-N,N-dimethyl-2H-tetrazol...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of CDK2/cyclin A2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM179929(US9133148, 1a)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of human MAGL transfected in human HEK293T cells assessed as reduction in ABPP binding by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  6nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563791(CHEMBL4778803)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563794(CHEMBL4793668)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50394389(CHEMBL2159798)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563792(CHEMBL4788586)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563793(CHEMBL4793997)
Affinity DataIC50:  9nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563790(CHEMBL4780294)
Affinity DataIC50:  9nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50394384(CHEMBL2159803)
Affinity DataIC50:  9nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50394371(CHEMBL2159779)
Affinity DataIC50:  9nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50049456(CHEMBL3318318)
Affinity DataIC50:  10nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50394383(CHEMBL2159804)
Affinity DataIC50:  12nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563801(CHEMBL4779678)
Affinity DataIC50:  16nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563802(CHEMBL4793265)
Affinity DataIC50:  17nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50414921(CHEMBL570812)
Affinity DataIC50:  20nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50414921(CHEMBL570812)
Affinity DataIC50:  20nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563803(CHEMBL4797565)
Affinity DataIC50:  22nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Jamia Hamdard

LigandPNGBDBM50320491(2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...)
Affinity DataIC50:  30nMpH: 7.4Assay Description:Xanthine oxidase (XO) assay of 2-(benzylamino)-4-methyl-1,3-thiazole-5-carboxylic acid derivatives 5a-p was evaluated using Bovine milk XO (grade 1, ...More data for this Ligand-Target Pair
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50394388(CHEMBL2159799)
Affinity DataIC50:  33nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50049457(CHEMBL3318317)
Affinity DataIC50:  39nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate substrate incubated for 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563795(CHEMBL4786239)
Affinity DataIC50:  68nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563785(CHEMBL4792393)
Affinity DataIC50:  74nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50432829(CHEMBL2171700)
Affinity DataIC50:  78nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563809(CHEMBL4794817)
Affinity DataIC50:  117nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563797(CHEMBL4777523)
Affinity DataIC50:  151nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563808(CHEMBL4793077)
Affinity DataIC50:  196nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563796(CHEMBL4780477)
Affinity DataIC50:  242nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563800(CHEMBL4776276)
Affinity DataIC50:  282nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50414921(CHEMBL570812)
Affinity DataIC50:  424nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563799(CHEMBL4785038)
Affinity DataIC50:  780nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563798(CHEMBL4800406)
Affinity DataIC50:  815nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563788(CHEMBL4798413)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Jamia Hamdard

LigandPNGBDBM178040(4-methyl-2-{[(2-methylphenyl)methyl]amino}-1,3-thi...)
Affinity DataIC50:  3.60E+3nMpH: 7.4Assay Description:Xanthine oxidase (XO) assay of 2-(benzylamino)-4-methyl-1,3-thiazole-5-carboxylic acid derivatives 5a-p was evaluated using Bovine milk XO (grade 1, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563787(CHEMBL4788417)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Jamia Hamdard

LigandPNGBDBM178041(2-{[(2,4-dichlorophenyl)methyl]amino}-4-methyl-1,3...)
Affinity DataIC50:  8.10E+3nMpH: 7.4Assay Description:Xanthine oxidase (XO) assay of 2-(benzylamino)-4-methyl-1,3-thiazole-5-carboxylic acid derivatives 5a-p was evaluated using Bovine milk XO (grade 1, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Jamia Hamdard

LigandPNGBDBM178039(2-{[(2-chlorophenyl)methyl]amino}-4-methyl-1,3-thi...)
Affinity DataIC50:  9.90E+3nMpH: 7.4Assay Description:Xanthine oxidase (XO) assay of 2-(benzylamino)-4-methyl-1,3-thiazole-5-carboxylic acid derivatives 5a-p was evaluated using Bovine milk XO (grade 1, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50401472(CHEMBL2204564)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human recombinant COX2 using PGG2 as substrate and N,N,N,N-tetramethyl-p-phenylnediamine measured for 25 secs by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Jamia Hamdard (Hamdard University)

Curated by ChEMBL
LigandPNGBDBM50401473(CHEMBL2204556)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of human recombinant COX2 using PGG2 as substrate and N,N,N,N-tetramethyl-p-phenylnediamine measured for 25 secs by spectrophotometric ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563786(CHEMBL4783652)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Jamia Hamdard

LigandPNGBDBM178043(2-{[(2-methoxyphenyl)methyl]amino}-4-methyl-1,3-th...)
Affinity DataIC50:  1.47E+4nMpH: 7.4Assay Description:Xanthine oxidase (XO) assay of 2-(benzylamino)-4-methyl-1,3-thiazole-5-carboxylic acid derivatives 5a-p was evaluated using Bovine milk XO (grade 1, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Jamia Hamdard

LigandPNGBDBM178036(2-{[(4-hydroxyphenyl)methyl]amino}-4-methyl-1,3-th...)
Affinity DataIC50:  2.15E+4nMpH: 7.4Assay Description:Xanthine oxidase (XO) assay of 2-(benzylamino)-4-methyl-1,3-thiazole-5-carboxylic acid derivatives 5a-p was evaluated using Bovine milk XO (grade 1, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563782(CHEMBL4786879)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50128581(Biphenyl-3-yl-carbamic acid cyclohexyl ester | CHE...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Jamia Hamdard

LigandPNGBDBM178033(2-{[(4-fluorophenyl)methyl]amino}-4-methyl-1,3-thi...)
Affinity DataIC50:  3.03E+4nMpH: 7.4Assay Description:Xanthine oxidase (XO) assay of 2-(benzylamino)-4-methyl-1,3-thiazole-5-carboxylic acid derivatives 5a-p was evaluated using Bovine milk XO (grade 1, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50274981(4-(4,5-dihydrothiazol-2-yl)phenyl butylcarbamate |...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563781(CHEMBL4800077)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetXanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Jamia Hamdard

LigandPNGBDBM178034(2-{[(4-bromophenyl)methyl]amino}-4-methyl-1,3-thia...)
Affinity DataIC50:  4.32E+4nMpH: 7.4Assay Description:Xanthine oxidase (XO) assay of 2-(benzylamino)-4-methyl-1,3-thiazole-5-carboxylic acid derivatives 5a-p was evaluated using Bovine milk XO (grade 1, ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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