Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM21216'
TargetAdenosine receptor A1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM21216(2-[4-(ethylsulfanyl)-1H-1,3-benzodiazol-2-yl]quino...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21216(2-[4-(ethylsulfanyl)-1H-1,3-benzodiazol-2-yl]quino...)
Affinity DataKi:  0.5nM ΔG°:  -53.1kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed