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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Ligand = 'BDBM50305817'
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50305817(1-(4-phenoxybenzyl)-5-(trifluoromethoxy)indoline-2...)
Affinity DataEC50:  1.90E+3nMAssay Description:Positive allosteric modulation activity at muscarinic M5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50305817(1-(4-phenoxybenzyl)-5-(trifluoromethoxy)indoline-2...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human muscarinic M5 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed