TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of California At San Diego
Curated by ChEMBL
University Of California At San Diego
Curated by ChEMBL
Affinity DataIC50: 0.0740nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Protein kinase C zetaMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C eta isozymeMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Protein kinase C beta 2More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C delta isozymeMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Mcgill University
Curated by ChEMBL
Mcgill University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of PKCeta (unknown origin) by IMAP kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of protein kinase C beta 1More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C epsilonMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C gammaMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C beta 2More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C beta 1 isozymeMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C epsilon isozymeMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C beta 2 isozymeMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C epsilonMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Protein kinase C gammaMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of Protein kinase C epsilonMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C gamma isozymeMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of Protein Kinase C etaMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of protein kinase C etaMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of protein kinase C epsilonMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of protein kinase C deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of protein kinase C gammaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of California At San Diego
Curated by ChEMBL
University Of California At San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of California At San Diego
Curated by ChEMBL
University Of California At San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of California At San Diego
Curated by ChEMBL
University Of California At San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Protein kinase C beta 2More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of protein kinase C beta IMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of California At San Diego
Curated by ChEMBL
University Of California At San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C alpha isozymeMore data for this Ligand-Target Pair