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Found 85 Enz. Inhib. hit(s) with Target = 'cAMP-dependent protein kinase catalytic subunit gamma'
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataKi:  4nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataKi:  170nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405349(CHEMBL5271837)
Affinity DataKi:  740nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405333(CHEMBL5270570)
Affinity DataKi:  744nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50216682(1-(5-Isoquinolinesulfonyl)-2-methylpiperazine | 1-...)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of ATP from protein kinase A (PKA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405348(CHEMBL5280643)
Affinity DataKi:  3.00E+3nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50223628(CHEMBL1161622)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of protein kinase A expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405346(CHEMBL5266306)
Affinity DataKi:  8.50E+4nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405336(CHEMBL5277116)
Affinity DataKi:  1.39E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405334(CHEMBL5280829)
Affinity DataKi:  1.55E+5nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405329(CHEMBL5279025)
Affinity DataKi:  1.74E+5nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405337(CHEMBL5268186)
Affinity DataKi:  3.54E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405328(CHEMBL5278563)
Affinity DataKi:  3.90E+5nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405341(CHEMBL5287370)
Affinity DataKi:  5.40E+5nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405343(CHEMBL5279009)
Affinity DataKi:  5.88E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405340(CHEMBL5276693)
Affinity DataKi:  9.55E+5nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405347(CHEMBL5281989)
Affinity DataKi:  1.42E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405342(CHEMBL5273882)
Affinity DataKi:  2.10E+6nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405344(CHEMBL5278260)
Affinity DataKi:  4.74E+6nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405331(CHEMBL5276685)
Affinity DataKi:  5.00E+6nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced platelet aggregation in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405338(CHEMBL2393369)
Affinity DataKi:  5.00E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405339(CHEMBL5286003)
Affinity DataKi:  6.22E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405345(CHEMBL5273503)
Affinity DataKi:  6.38E+6nMAssay Description:In vitro inhibition of angiotensin converting enzyme isolated from rat lung.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405332(CHEMBL5285449)
Affinity DataKi:  1.00E+7nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50405335(CHEMBL2357735)
Affinity DataKi:  2.00E+7nMAssay Description:In vitro inhibition of Neutral Endopeptidase isolated from rat kidney.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50: <1nMAssay Description:Inhibition of PKA (unknown origin) after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human PKAcg using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50587770(CHEMBL5188493)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228843(CHEMBL436718)
Affinity DataIC50:  3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM3149(2-{[2,6-dihydroxy-4-({[(3R,4R)-3-[(4-hydroxybenzen...)
Affinity DataIC50:  4nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  6.5nMAssay Description:In vitro inhibition of Protein Kinase AMore data for this Ligand-Target Pair
In DepthDetails
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of human PKAcg using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50242733(AT-13148)
Affinity DataIC50: <10nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM15211(CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...)
Affinity DataIC50:  50nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50587769(CHEMBL5181354)
Affinity DataIC50:  159nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50614310(CHEMBL5269663)
Affinity DataIC50:  184nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50280450(18-hydroxy-3-methoxy-2-methyl-4-methylamino-(2R,3S...)
Affinity DataIC50:  250nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50280450(18-hydroxy-3-methoxy-2-methyl-4-methylamino-(2R,3S...)
Affinity DataIC50:  250nMAssay Description:Inhibition of protein kinase AMore data for this Ligand-Target Pair
In DepthDetails
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228839(CHEMBL415414)
Affinity DataIC50:  300nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50506921(CHEMBL4459800)
Affinity DataIC50:  790nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228838(CHEMBL428973)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM15211(CHEMBL104264 | H-89 | H89 | HT-89 (H-89) | N-(2-{[...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of PKA-mediated phosphorylation of kemptide at 100 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228847(CHEMBL407100)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50228846(CHEMBL265876)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50358686(CHEMBL1922138)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50614312(CHEMBL5284365)
Affinity DataIC50:  1.52E+3nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50614314(CHEMBL5269818)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of PKA (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
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