Found 76 of ic50 for monomerid = 50001683 
Affinity DataIC50: 0.140nMAssay Description:Agonist activity at delta opioid expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulationMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:Binding affinity against rat Opioid receptor delta 1 expressed in CHO cells determined by competitive inhibition of 1 nM [3H]DPDPE.More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Agonist activity at human delta opioid receptor expressed in HEK293 cells assessed as inhibition of forskolin-induced cAMP production after 30 mins b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Compound was evaluated for the binding affinity in comparison with [3H]-[p-Cl-Phe4]-DPDPE (opioid receptor delta selective ligand)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration was determined against delta-opioid receptor using [3H]- DPDPE radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Tested for inhibitory concentration against [3H]DPDPE binding at sites of delta-opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Tested for the binding affinity against the Kappa opioid receptor in guinea pig brain using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibitory potency against Opioid receptor delta 1 was determined in electrically induced smooth muscle contractions of mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Compound is tested in vitro in mouse vas deferens (MVD) assay mediated by Opioid receptor delta 1More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Compound was tested for agonistic activity against the opioid receptor in electrically stimulated mouse vas deference.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding potency of compound in competition with [3H]DPDPE for Opioid receptor delta 1 tested in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibitory activity measured against Opioid receptor delta 1 using mouse vas deference assay (MVD).More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Compound was evaluated for its inhibitory potency against opioid receptor delta of Mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Ability to inhibit electrically evoked contractions of isolated muscle preparations of mouse vas deference (MVD, delta receptor)More data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Opioid activity against delta-receptor of isolated mouse vas deferens(MVD) at 30 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Agonistic activity towards Opioid receptor delta 1 as inhibitory activity towards electrically stimulated mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Agonist activity was evaluated in guinea pig ileum (GPI) preparations at Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Tested for agonist activity against delta opioid receptor mouse vas deferensMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Ability to displace [3H]DPDPE from Opioid receptor delta 1 in rat brain membranes, was determined from radioreceptor assay.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Opioid receptor binding affinity in rat brain membrane preparations by the displacement of [3H]DSLET (Opioid receptor delta 1-selective radioligand)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibitory activity measured against [3H]DPDPE (Opioid receptor delta 1 ligand) in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Binding affinity towards delta opioid receptor was determined in rat brain using [H]-[p-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80nMAssay Description:Inhibitory concentration required for 50 percent inhibition of opioid receptor delta 1 induced contractions in mouse vas deferens (MVD) smooth muscle...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Compound was evaluated for the binding affinity in comparison with [3H]- DPDPE (opioid receptor delta selective ligand)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of binding of radioligand [3H][p-Cl-phe]-DPDPE to Opioid receptor delta 1 in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 385nMAssay Description:The ability to displace [3H]naloxone from the Opioid receptor mu 1 isolated from rat brain membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 609nMAssay Description:Binding affinity opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 609nMAssay Description:Compound was evaluated for its ability to displace [3H]- CTOP (opioid receptor mu selective ligand)More data for this Ligand-Target Pair
Affinity DataIC50: 609nMAssay Description:Ability to displace [3H]CTOP from Opioid receptor mu 1 in rat brain membranes, was determined from radioreceptor assayMore data for this Ligand-Target Pair
Affinity DataIC50: 609nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]- CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 619nMAssay Description:Inhibitory activity measured against [3H]CTOP (Opioid receptor mu 1) in rat brain using radioreceptor binding assays.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Institute For Bioorganic Research
Curated by ChEMBL
Institute For Bioorganic Research
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Inhibitory concentration against delta opioid receptor of electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Binding affinity towards mu opioid receptor was determined in rat brain using [3H]CTOP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Tested for inhibitory concentration against [3H]DAMGO binding at sites of mu-opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration was determined against Opioid receptor mu 1 using [3H]- DAMGO radioligandMore data for this Ligand-Target Pair
