TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
University Of Eastern Piedmont
Curated by ChEMBL
University Of Eastern Piedmont
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Antagonist activity at recombinant rat TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced intracellular calcium level incubated...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Agonist activity at TRPA1 (unknown origin) channel desensitization in presence of icilinMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Agonist activity at TRPA1 (unknown origin) channel desensitization in presence of isothiocyanateMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) channel desensitization in presence of 4alphaPDDMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 3(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 9.40E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV3 (unknown origin) channel desensitization in presence of carvacrolMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Homo sapiens)
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 1.57E+4nMAssay Description:Agonist activity at ionomycin-stimulated TRPV2 (unknown origin) channel desensitization in presence of lysophosphatidylcholineMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Non competitive inhibition of CYP2J2 (unknown origin) in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.04E+4nMAssay Description:Non competitive inhibition of recombinant human CYP2A6 using coumarin as substrate preincubated with NADPH for 20 mins and measured after 30 minMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of FAAH in rat brain membranes using [14C]-AEA as substrate measured after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human DAGLalpha expressed in COS7 cells using [14C]-oleoyl-2-arachidonoyl-glycerol as substrate measured after 20 mins by b...More data for this Ligand-Target Pair
TargetN-acylethanolamine-hydrolyzing acid amidase(Homo sapiens (Human))
Concordia University Wisconsin
Curated by ChEMBL
Concordia University Wisconsin
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human NAAA expressed in HEK293 cells using [14C]-N-palmitoylethanolamine as substrate measured after 30 mins by beta-counti...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 8.20E+4nMAssay Description:Agonist activity at ionomycin-stimulated TRPV1 (unknown origin) channel desensitization in presence of capsaicinMore data for this Ligand-Target Pair