Found 3 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 4' and Ligand = 'BDBM50061117'
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) channel desensitization in presence of 4alphaPDDMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rattus norvegicus)
University Of Eastern Piedmont
Curated by ChEMBL
University Of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.61E+4nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataEC50: 1.61E+4nMAssay Description:Agonist activity at ionomycin-stimulated TRPV4 (unknown origin) activationMore data for this Ligand-Target Pair