Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Binding affinity for Adenosine A2A receptor from rat striatal membranes using [3H]-CGH 21680More data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 4.77nMAssay Description:Binding affinity for Adenosine A2A receptor from rat striatal membranes using [3H]-CGH 21680More data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 7.05nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at rat adenosine 2A receptor assessed as reduction in cAMP level in presence of 0.1 uM adenosineMore data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
Affinity DataIC50: >10nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Activity at adenosine A2A receptor in rat PC12 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity for Adenosine A2A receptor using [3H]-ZM-241,38 in ratMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Activity at adenosine A2A receptor in rat PC12 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Activity at adenosine A2A receptor in rat PC12 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 66.9nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Binding affinity against Adenosine A2A receptor in rat striatal membranes b displacement of [3H]-CGS- 21680More data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Antagonist activity at rat adenosine 2A receptor assessed as reduction in cAMP level in presence of 10 uM adenosineMore data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Binding affinity for Adenosine A2A receptor from rat striatal membranes using [3H]-CGH 21680More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 228nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptor in presence of 100 mM NaClMore data for this Ligand-Target Pair
Affinity DataIC50: 263nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 366nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptor in presence of 100 mM NaClMore data for this Ligand-Target Pair
Affinity DataIC50: 531nMAssay Description:Binding affinity for Adenosine A2A receptor from rat striatal membranes using [3H]-CGH 21680More data for this Ligand-Target Pair
Affinity DataIC50: 750nMAssay Description:Antagonist activity at recombinant rat A2A adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 840nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.66E+3nMAssay Description:Binding affinity to adenosine A2A receptor in rat brain striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]-NECA in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair