Report error Found 93 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM21220'
Affinity DataEC50: 394nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
Affinity DataEC50: 394nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:G-protein activation in human Adenosine A2A receptor expressing CHO cells using cAMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Potency against cAMP formation in CHO cells expressing recombinant human A2A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 394nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 34nMAssay Description:Efficacy against phenylephrine precontracted tissue relaxation in rat aortaMore data for this Ligand-Target Pair
Affinity DataEC50: 21.9nMAssay Description:Agonist activity at human adenosine A2A receptor expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Agonist activity at human recombinant adenosine A2A receptor expressed in CHO cells assessed as [3H]cAMP accumulation after 15 mins by liquid scintil...More data for this Ligand-Target Pair
Affinity DataEC50: 17.6nMAssay Description:Agonist activity at human adenosine A2A receptor expressed in CHO-K1 cells by cAMP accumulation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist activity at human adenosine A2A receptor expressed in CHO cells assessed as stimulation of [3H]cAMP levels by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Agonist activity at human A2A-AR expressed in FlpIn-CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation preincubated for 40 mi...More data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Agonist activity at Homo sapiens (human) adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.5nMAssay Description:Irreversible agonist activity at human adenosine A2A receptor expressed in Flp-In-CHO cells assessed as effect on forskolin-induced cAMP accumulation...More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human adenosine A2A receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated fo...More data for this Ligand-Target Pair
Affinity DataEC50: 4.80nMAssay Description:Agonist activity at human A2A receptor expressed in Flp-In-CHO cells assessed as cAMP accumulation incubated for 30 mins by LANCE cAMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 339nMAssay Description:Agonist activity at human Adenosine A2A receptor expressed in yeast cells coexpressed with chimeric GPA1/Galphas after 16 hrs by beta-galactosidase r...More data for this Ligand-Target Pair
Affinity DataIC50: 7.05nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Agonist activity at adenosine A2A receptor in human neutrophils assessed as inhibition of fMLP-induced reactive oxygen species release by chemilumine...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]CGS 21680 from human recombinant adenosine receptor A2A expressed in HEK293 cells measured after 120 mins by scintillation counti...More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]CGS 21680 from human recombinant adenosine A2a receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of human adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 366nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptor in presence of 100 mM NaClMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro inhibition of human neutrophil activation via Adenosine A2A receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity against Q89D human adenosine A2A receptor expressed in CHO cells using [3H]- ZM-241385 More data for this Ligand-Target Pair
Affinity DataKi: 1.5nM ΔG°: -50.4kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity to A2A adenosine receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity of ligand at human adenosine receptors expressed in CHO cell. More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity to human A2A adenosine receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.13nMAssay Description:Binding affinity for Adenosine A2A receptor in rat brain membranes using [3H]CGS-21680 More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Binding affinity for HA-tagged mutant human Adenosine A2A receptor (H250N) using [3H]-CGS-21,680 as radioligand expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity against adenosine A2a receptor from rat striatum using [3H]-CGS- 21680 as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H]-CGS- 51680 from Adenosine A2A receptor of rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptor expressed in CHO cell membranes incubated for 120 mins by scintillation counting metho...More data for this Ligand-Target Pair
Affinity DataKi: 9.30nM ΔG°: -45.8kJ/molepH: 7.4 T: 2°CAssay Description:Binding affinity of ligand at WT and mutant human A2A ARs expressed in COS7 cell. More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to adenosine A2A receptor in rat striatal membranes by measuring displacement of specific [3H]-CGS- 21680 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3 H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from rat adenosine receptor A2A after 60 mins by liquid s...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against adenosine A1 receptor from rat brain membranes using [3H]cyclohexyladenosine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against adenosine A2A receptor in rat striatal membranes using [3H]-CGS- 21680.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of [3H]- CGS 21680 binding to Adenosine A2A receptor of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from rat A2A adenosine receptor expressed in HEK293 cell mem...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of 3[H]CGS21680 from rat A2A adenosine receptor expressed in HEK293 cells after 60 min by Liquid scintillation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 12.2nMAssay Description:Displacement of [3H]CGS-21680 binding to Adenosine A2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12.4nMAssay Description:Binding affinity towards adenosine A2A receptor in rat brain striatumMore data for this Ligand-Target Pair
Affinity DataKi: 12.4nMAssay Description:Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12.5nMAssay Description:Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
