Compile Data Set for Download or QSAR
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Found 5 of ic50 for UniProtKB: A0A024RBH0
TargetCyclin-Y/Cyclin-dependent kinase 17(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  10.7nMAssay Description:Inhibition of human CDK17/cyclin-Y using MBP protein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-Y/Cyclin-dependent kinase 17(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  16.3nMAssay Description:Inhibition of human CDK17/cyclin-Y using MBP protein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 17(Homo sapiens (Human))TBA
LigandPNGBDBM50404389(CHEMBL5285499)
Affinity DataIC50: >1.20E+3nMAssay Description:Displacement of specifically bound [3H]naloxone from rat brain homogenate, in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails
TargetCyclin-dependent kinase 17(Homo sapiens (Human))TBA
LigandPNGBDBM50593922(CHEMBL5199065)
Affinity DataIC50: >1.20E+3nMAssay Description:Displacement of specifically bound [3H]naloxone from rat brain homogenate, in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails
TargetCyclin-dependent kinase 17(Homo sapiens (Human))TBA
LigandPNGBDBM126500(US11591322, Compound NVP-2 | US8778951, 310)
Affinity DataIC50:  1.50E+3nMAssay Description:Effective concentration required for inhibitory activity towards human beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails