TargetCyclin-Y/Cyclin-dependent kinase 17(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 10.7nMAssay Description:Inhibition of human CDK17/cyclin-Y using MBP protein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCyclin-Y/Cyclin-dependent kinase 17(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 16.3nMAssay Description:Inhibition of human CDK17/cyclin-Y using MBP protein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+3nMAssay Description:Displacement of specifically bound [3H]naloxone from rat brain homogenate, in the absence of NaClMore data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+3nMAssay Description:Displacement of specifically bound [3H]naloxone from rat brain homogenate, in the absence of NaClMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Effective concentration required for inhibitory activity towards human beta-1 adrenergic receptorMore data for this Ligand-Target Pair