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Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50046853
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7398((2 Z)-6 -Bromoindirubin | 6 -bromoindirubin | 6-br...)
Affinity DataIC50:  4nMAssay Description:Competitive inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 30 mins by scintillation counting analysis i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7287(8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,17}]octad...)
Affinity DataIC50:  4nMAssay Description:Competitive inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 30 mins by scintillation counting analysis i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7262(14-nitro-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,...)
Affinity DataIC50:  5nMAssay Description:Inhibition of glycogen synthase kinase-3 (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7463(4,5-diphenyl-1H-pyrazolo[3,4-c]pyridazin-3-amine |...)
Affinity DataIC50:  250nMAssay Description:Inhibition of glycogen synthase kinase-3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM50135214(CHEMBL3747661)
Affinity DataIC50:  400nMAssay Description:Competitive inhibition of glycogen synthase kinase-3 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7876(2-bromo-1-(4-bromophenyl)ethan-1-one | Halomethyl ...)
Affinity DataIC50:  500nMAssay Description:Inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 20 mins by scintillation counting analysis in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7877(2-bromo-1-(4-chlorophenyl)ethan-1-one | Halomethyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 20 mins by scintillation counting analysis in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM50135211(CHEMBL3747426)
Affinity DataIC50:  1.28E+3nMAssay Description:Inhibition of glycogen synthase kinase-3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM50119691(2-Bromo-1-(4-nitro-phenyl)-ethanone | CHEMBL106072)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 20 mins by scintillation counting analysis in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7874(2-chloro-1-(4-chlorophenyl)ethan-1-one | Halomethy...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 20 mins by scintillation counting analysis in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7875(2-bromo-1-phenylethan-1-one | CHEMBL102953 | Halom...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 20 mins by scintillation counting analysis in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM50135212(CHEMBL3746095)
Affinity DataIC50:  7.05E+3nMAssay Description:Inhibition of glycogen synthase kinase-3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM7873(2-chloro-1-phenylethan-1-one | CHEMBL105712 | Halo...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 20 mins by scintillation counting analysis in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Central University

Curated by ChEMBL
LigandPNGBDBM50134240(CHEMBL3745772)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of glycogen synthase kinase-3 beta (unknown origin) using GS-1 as substrate after 20 mins by scintillation counting analysis in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed