Reaction Details Report a problem with these data
Target
Regulatory protein E2
Ligand
BDBM50035218
Substrate
n/a
Meas. Tech.
ChEMBL_532975 (CHEMBL989645)
Kd
>400000±n/a nM
Citation
Saitoh, T; Kuramochi, K; Imai, T; Takata, K; Takehara, M; Kobayashi, S; Sakaguchi, K; Sugawara, F Podophyllotoxin directly binds a hinge domain in E2 of HPV and inhibits an E2/E7 interaction in vitro. Bioorg Med Chem 16:5815-25 (2008) [PubMed] Article
More Info.:
Target
Name:
Regulatory protein E2
Synonyms:
E2 | VE2_HPV1
Type:
PROTEIN
Mol. Mass.:
45494.82
Organism:
Human papillomavirus type 1a
Description:
ChEMBL_532977
Residue:
401
Sequence:
MENLSSRLDLLQEQLMNLYEQDSKLIEDQIKQWNLIRQEQVLFHFARKNGVMRIGLQAVPSLASSQEKAKTAIEMVLHLESLKDSPYGTEDWSLQDTSRELFLAPPAGTFKKSGSTLEVTYDNNPDNQTRHTIWNHVYYQNGDDVWRKVSSGVDAVGVYYLEHDGYKNYYVLFAEEASKYSTTGQYAVNYRGKRFTNVMSSTSSPRAAGAPAVHSDYPTLSESDTAQQSTSIDYTELPGQGETSQVRQRQQKTPVRRRPYGRRRSRSPRGGGRREGESTPSRTPGSVPSARDVGSIHTTPQKGHSSRLRRLLQEAWDPPVVCVKGGANQLKCLRYRLKASTQVDFDSISTTWHWTDRKNTERIGSARMLVKFIDEAQREKFLERVALPRSVSVFLGQFNGS