Reaction Details Report a problem with these data
Target
Beta-2-microglobulin
Ligand
BDBM92397
Substrate
n/a
Meas. Tech.
Fluorescence Assay
pH
7.4±0
Temperature
310.15±0 K
IC50
4.9e+4± 9e+3 nM
Citation
Giorgetti, S; Raimondi, S; Pagano, K; Relini, A; Bucciantini, M; Corazza, A; Fogolari, F; Codutti, L; Salmona, M; Mangione, P; Colombo, L; De Luigi, A; Porcari, R; Gliozzi, A; Stefani, M; Esposito, G; Bellotti, V; Stoppini, M Effect of tetracyclines on the dynamics of formation and destructuration of beta2-microglobulin amyloid fibrils. J Biol Chem 286:2121-31 (2011) [PubMed] Article
More Info.:
Target
Name:
Beta-2-microglobulin
Synonyms:
B2M | B2MG_HUMAN
Type:
Enzyme
Mol. Mass.:
13714.40
Organism:
Homo sapiens (Human)
Description:
P61769
Residue:
119
Sequence:
MSRSVALAVLALLSLSGLEAIQRTPKIQVYSRHPAENGKSNFLNCYVSGFHPSDIEVDLLKNGERIEKVEHSDLSFSKDWSFYLLYYTEFTPTEKDEYACRVNHVTLSQPKIVKWDRDM