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Found 159 with Last Name = 'stefani' and Initial = 'm'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50081081(6-{4-[2-(4-Quinolin-8-yl-piperazin-1-yl)-ethyl]-ph...)
Affinity DataKi:  3nMAssay Description:Binding affinity of compound to human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50081081(6-{4-[2-(4-Quinolin-8-yl-piperazin-1-yl)-ethyl]-ph...)
Affinity DataKi:  11nMAssay Description:Binding ability of compound to human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50081081(6-{4-[2-(4-Quinolin-8-yl-piperazin-1-yl)-ethyl]-ph...)
Affinity DataKi:  14nMAssay Description:Binding affinity of compound to human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50081082(2-(4-{2-[4-(6-Amino-pyridin-2-yl)-phenyl]-ethyl}-p...)
Affinity DataKi:  320nMAssay Description:Binding affinity of compound to m2 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50081082(2-(4-{2-[4-(6-Amino-pyridin-2-yl)-phenyl]-ethyl}-p...)
Affinity DataKi:  590nMAssay Description:Binding ability of compound to m4 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033236(8,9-Dichloro-2-methyl-5-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50:  0.300nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033242(3-Cyclohexyl-6-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.400nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033257(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  0.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033238(3-(4-Chloro-phenyl)-1,8-dimethyl-5-[4-(2-methyl-im...)
Affinity DataIC50:  0.600nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033240(1-Methyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  0.600nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033264(3-Cyclohexyl-1,8-dimethyl-5-[4-(2-methyl-imidazo[4...)
Affinity DataIC50:  0.700nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033260(3-Isobutoxymethyl-1,8-dimethyl-5-[4-(2-methyl-imid...)
Affinity DataIC50:  0.800nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033234(1,3-Dimethyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033233(8,9-Dichloro-1-methyl-5-[4-(2-methyl-imidazo[4,5-c...)
Affinity DataIC50:  1.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033249(5,7,9-Trimethyl-2-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  1.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033229(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033245(8-Bromo-5-methyl-2-[4-(2-methyl-imidazo[4,5-c]pyri...)
Affinity DataIC50:  1.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033255(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033232(8,9-Dichloro-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  1.70nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033263(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  2.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033251(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  2.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033231(1,8,9-Trimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  2.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033246(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  2.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033243(1-Methyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  2.70nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033230(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  3.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033268(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)
Affinity DataIC50:  3.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033241(3-Isopropyl-1,8-dimethyl-5-[4-(2-methyl-imidazo[4,...)
Affinity DataIC50:  3.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033254(8-Bromo-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl)...)
Affinity DataIC50:  4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033235(7-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)
Affinity DataIC50:  4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033239(8-Bromo-1-methyl-4-[4-(2-methyl-imidazo[4,5-c]pyri...)
Affinity DataIC50:  4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)
Affinity DataIC50:  4.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033266(1,3,4-Trimethyl-7-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033237(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  5.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033267(8-Bromo-4-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl)...)
Affinity DataIC50:  5.60nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMisshapen-like kinase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50361467(CHEMBL1938400)
Affinity DataIC50:  6nMAssay Description:Inhibition of MINKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033253(3-(2-Methoxy-ethoxymethyl)-1,8-dimethyl-5-[4-(2-me...)
Affinity DataIC50:  6.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033258(7,9-Dimethyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  6.80nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033248(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  11nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033261(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  14nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033256(3-Hydroxymethyl-1,8-dimethyl-5-[4-(2-methyl-imidaz...)
Affinity DataIC50:  14nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50072197(2-[4-(3,5-Bis-cyclopropylmethoxy-phenyl)-2-ethyl-6...)
Affinity DataIC50:  15nMAssay Description:Evaluated for the inhibition of [3H]rolipram binding to membrane-bound PDE4.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50072197(2-[4-(3,5-Bis-cyclopropylmethoxy-phenyl)-2-ethyl-6...)
Affinity DataIC50:  16nMAssay Description:Evaluated for its ability to inhibit PDE3.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033228(1,3,8-Trimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  17nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033227(7,9-Dimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  21nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4D(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50072197(2-[4-(3,5-Bis-cyclopropylmethoxy-phenyl)-2-ethyl-6...)
Affinity DataIC50:  22nMAssay Description:Evaluated for its ability to inhibit PDE4D.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50361467(CHEMBL1938400)
Affinity DataIC50:  23nMAssay Description:Inhibition of p38beta MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(RAT)
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50072197(2-[4-(3,5-Bis-cyclopropylmethoxy-phenyl)-2-ethyl-6...)
Affinity DataIC50:  25nMAssay Description:Evaluated for its ability to inhibit PDE4B.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033262(1,3-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)
Affinity DataIC50:  26nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A(Homo sapiens (Human))
Novartis Pharma

Curated by ChEMBL
LigandPNGBDBM50072197(2-[4-(3,5-Bis-cyclopropylmethoxy-phenyl)-2-ethyl-6...)
Affinity DataIC50:  30nMAssay Description:Evaluated for its ability to inhibit PDE4A.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50033247(1,7,9-Trimethyl-4-[4-(2-methyl-imidazo[4,5-c]pyrid...)
Affinity DataIC50:  38nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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