Compile Data Set for Download or QSAR
Report error Found 138 of affinity data for UniProtKB/TrEMBL: P00761
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425657(CHEMBL2315245)
Affinity DataKi:  0.600nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425656(CHEMBL2315246)
Affinity DataKi:  3nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425661(CHEMBL2315240)
Affinity DataKi:  3.40nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425659(CHEMBL2315242)
Affinity DataKi:  7.80nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425655(CHEMBL2315247)
Affinity DataKi:  10nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532391(CHEMBL4591922)
Affinity DataKi:  14nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532391(CHEMBL4591922)
Affinity DataKi:  14nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425652(CHEMBL2315234)
Affinity DataKi:  18nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425654(CHEMBL2315236)
Affinity DataKi:  18nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425660(CHEMBL2315241)
Affinity DataKi:  19nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532389(CHEMBL4458743)
Affinity DataKi:  21nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532389(CHEMBL4458743)
Affinity DataKi:  21nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425658(CHEMBL2315244)
Affinity DataKi:  25nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157098(6-[2-((S)-1-Isopropyl-3,4-dihydro-isoquinolin-7-yl...)
Affinity DataKi:  30nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157093(6-[2-(1-Cyclohexyl-2-methyl-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  31nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425648(CHEMBL2315243)
Affinity DataKi:  38nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50147096(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)
Affinity DataKi:  40nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425653(CHEMBL2315237)
Affinity DataKi:  42nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50147088(6-Carbamimidoyl-4-furan-3-yl-naphthalene-2-carboxy...)
Affinity DataKi:  45nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157096(6-[2-(1-Isopropyl-3,4-dihydro-isoquinolin-7-yl)-cy...)
Affinity DataKi:  53nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157087(6-(2-phenylcyclopropyl)-8-(pyrimidin-2-ylamino)-2-...)
Affinity DataKi:  54nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425651(CHEMBL2315235)
Affinity DataKi:  55nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532387(CHEMBL4476141)
Affinity DataKi:  62nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532387(CHEMBL4476141)
Affinity DataKi:  62nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425649(CHEMBL2315239)
Affinity DataKi:  63nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157099(4-Bromo-6-carbamimidoyl-naphthalene-2-carboxylic a...)
Affinity DataKi:  64nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157094(8-(Pyrimidin-2-ylamino)-6-((E)-styryl)-naphthalene...)
Affinity DataKi:  84nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157090(6-(2-(1-isopropyl-2-methyl-1,2,3,4-tetrahydroisoqu...)
Affinity DataKi:  90nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157084(8-Furan-3-yl-6-styryl-naphthalene-2-carboxamidine ...)
Affinity DataKi:  96nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50044092(spumigin E)
Affinity DataIC50: 100nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532406(CHEMBL4545331)
Affinity DataKi:  103nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532406(CHEMBL4545331)
Affinity DataKi:  103nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532401(CHEMBL4515955)
Affinity DataKi:  109nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532401(CHEMBL4515955)
Affinity DataKi:  109nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50425650(CHEMBL2315238)
Affinity DataKi:  126nMAssay Description:Inhibition of pig trypsin using CH3SO2-D-Cha-Gly-Arg-pNA as substrate after 5 to 10 mins by micro plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50080139((R)-2-({5-[(S)-1-((R)-1-Carboxy-ethylcarbamoyl)-et...)
Affinity DataKi:  128nMAssay Description:Inhibition constant (Ki) when mixed with p-nitroanilide against trypsin enzyme for the conversion of water-soluble compound to fluorescent oil-solubl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50080139((R)-2-({5-[(S)-1-((R)-1-Carboxy-ethylcarbamoyl)-et...)
Affinity DataKi:  128nMAssay Description:Inhibition constant (Ki) against trypsin enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532398(CHEMBL4454130)
Affinity DataKi:  136nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532398(CHEMBL4454130)
Affinity DataKi:  136nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157088(6-[2-(3-Isopropoxy-phenyl)-cyclopropyl]-naphthalen...)
Affinity DataKi:  141nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532392(CHEMBL4437656)
Affinity DataKi:  156nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532392(CHEMBL4437656)
Affinity DataKi:  156nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157097(6-[2-(1-Phenyl-3,4-dihydro-isoquinolin-7-yl)-cyclo...)
Affinity DataKi:  165nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157083(6-Phenethyl-8-(pyrimidin-2-ylamino)-naphthalene-2-...)
Affinity DataKi:  167nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50286441(Ac-LLR-CHO | Ac-Leu-Leu-Arg-H | (S)-2-((S)-2-Acety...)
Affinity DataIC50: 200nMAssay Description:Inhibition of pig pancreas trypsin type IX-SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50138670(uPa_7 | 6-carbamimidoyl-N-phenyl-2-naphthamide | 6...)
Affinity DataKi:  325nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157089(8-Bromo-6-(2-phenyl-cyclopropyl)-naphthalene-2-car...)
Affinity DataKi:  334nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50157082(6-Styryl-naphthalene-2-carboxamidine | CHEMBL18534...)
Affinity DataKi:  346nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50044094(CHEMBL3325623)
Affinity DataIC50: 350nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2016
Entry Details Article
PubMed
TargetTrypsin(Pig)
Philipps University Marburg

Curated by ChEMBL
LigandPNGBDBM50532394(CHEMBL4553652)
Affinity DataKi:  351nMAssay Description:Inhibition of porcine trypsin using Mes-DArg-Gly-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
Displayed 1 to 50 (of 138 total ) | Next | Last >>
Jump to: