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TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 0.354nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50225314(CHEMBL1627822)
Affinity DataKd:  0.620nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50148732(17alpha-ethinyl-19-nortestosterone | 17alpha-ethin...)
Affinity DataKd:  0.630nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM19441(Evista | CHEMBL81 | Keoxifene | Raloxifene, 6 | RA...)
Affinity DataIC50: 0.700nMAssay Description:Binding affinity for Rat Estrogen receptor-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50009716(Compound 133314 | TRIOXIFENE MESYLATE)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [2,4,6,7-3H]-estradiol from estrogen receptor in immature rat uterine cytosol by dextran-coated charcoal-adsorption assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50123209(5'-(2-hexahydro-1-pyridinylethoxy)-2-(4-hydroxyphe...)
Affinity DataIC50: 1.70nMAssay Description:Binding affinity for Rat Estrogen receptor-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]- Estradiol from Estrogen receptor of rat uterine cytosolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM19441(Evista | CHEMBL81 | Keoxifene | Raloxifene, 6 | RA...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 2nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50214281(MESO-HEXESTROL | Hexestrol)
Affinity DataIC50: 2nMAssay Description:Binding affinity for rat estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2018
Entry Details

TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50123208(2-(4-hydroxyphenyl)-3-methyl-1,2'-spirobi[1H-inden...)
Affinity DataIC50: 2.20nMAssay Description:Binding affinity for Rat Estrogen receptor-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50227469(CHEMBL285536)
Affinity DataEC50:  2.90nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50023749(4-[1-(4-hydroxyphenyl)-2-phenylvinyl]phenol | 4-(1...)
Affinity DataEC50:  3.20nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50227471(CHEMBL287352)
Affinity DataEC50:  3.30nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM8903(CHEMBL103 | (1S,2R,10S,11S,14S,15S)-14-acetyl-2,15...)
Affinity DataKd:  3.90nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50227470(CHEMBL34648)
Affinity DataEC50:  4.5nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataEC50:  5.70nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169743(CHEMBL1358 | (7R,8R,9S,13S,14S,17S)-13-methyl-7-(9...)
Affinity DataIC50: 5.89nMAssay Description:Displacement of [3H]estradiol from rat uterine cytosolic estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM20608([3H]4-OHT | cid_449459 | CHEMBL489 | AFIMOXIFENE |...)
Affinity DataEC50:  6nMAssay Description:In vitro displacement of 3 nM [3H]4-hydroxytamoxifen from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM19441(Evista | CHEMBL81 | Keoxifene | Raloxifene, 6 | RA...)
Affinity DataIC50: 7nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50054811({4-[(Z)-1-(4-Hydroxy-phenyl)-2-phenyl-but-1-enyl]-...)
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]- Estradiol from Estrogen receptor of rat uterine cytosolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50227471(CHEMBL287352)
Affinity DataEC50:  9.5nMAssay Description:In vitro displacement of 3 nM [3H]4-hydroxytamoxifen from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50471710(CHEMBL317748)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50227468(CHEMBL33879)
Affinity DataEC50:  10nMAssay Description:In vitro displacement of [3H]estradiol from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM20606((5R,6S)-6-phenyl-5-[4-(2-pyrrolidin-1-ylethoxy)phe...)
Affinity DataIC50: 11nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50471711(CHEMBL98892)
Affinity DataIC50: 11nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM20606((5R,6S)-6-phenyl-5-[4-(2-pyrrolidin-1-ylethoxy)phe...)
Affinity DataIC50: 11nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM86690(A-348441 | A 348441)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50123207(2-(3-hydroxyphenyl)-1,2'-spirobi[1H-indene]-6-ol |...)
Affinity DataIC50: 16nMAssay Description:Binding affinity for Rat Estrogen receptor-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118989((2-Chloro-phenyl)-(6-hydroxy-3-naphthalen-1-yl-ben...)
Affinity DataIC50: 30nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50123206(2-(3-hydroxyphenyl)-1,2'-spirobi[1H-indene]-5-ol |...)
Affinity DataIC50: 34nMAssay Description:Binding affinity for Rat Estrogen receptor-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50065941(1-{2-[4-(6-Methoxy-2-phenyl-3,4-dihydro-naphthalen...)
Affinity DataIC50: 41nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50471707(CHEMBL98116)
Affinity DataIC50: 47nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118987((2,4-Dimethyl-phenyl)-(6-hydroxy-3-naphthalen-1-yl...)
Affinity DataIC50: 75nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50119003(Biphenyl-4-yl-(6-hydroxy-3-naphthalen-1-yl-benzofu...)
Affinity DataIC50: 99nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50123212(2-phenyl-1,2'-spirobi[1H-indene]-5'-ol | CHEMBL439...)
Affinity DataIC50: 114nMAssay Description:Binding affinity for Rat Estrogen receptor-alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50154088(7-bromo-2-(4-hydroxyphenyl)benzo[d]oxazol-5-ol | 7...)
Affinity DataIC50: 132nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50471709(CHEMBL421389)
Affinity DataIC50: 132nMAssay Description:Inhibition of estradiol binding to estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50119000((2,3-Dihydro-benzo[1,4]dioxin-6-yl)-(6-hydroxy-3-n...)
Affinity DataIC50: 140nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118999((6-Hydroxy-3-naphthalen-1-yl-benzofuran-2-yl)-phen...)
Affinity DataIC50: 150nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50225310(CHEMBL1794824)
Affinity DataKd:  160nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50227469(CHEMBL285536)
Affinity DataEC50:  170nMAssay Description:In vitro displacement of 3 nM [3H]4-hydroxytamoxifen from estrogen receptor of rat uterine cystolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2019
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50154084(7-bromo-2-(3-fluoro-4-hydroxyphenyl)benzo[d]oxazol...)
Affinity DataIC50: 171nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118993((6-Hydroxy-3-naphthalen-1-yl-benzofuran-2-yl)-(4-h...)
Affinity DataIC50: 180nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50119006((3,4-Dihydro-2H-benzo[b][1,4]dioxepin-7-yl)-(6-hyd...)
Affinity DataIC50: 190nMAssay Description:Binding affinity for Estrogen receptor alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM86689(CAS_84371-65-3 | NSC_55245 | RU-486)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2017
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50119004((3-Fluoro-phenyl)-(6-hydroxy-3-naphthalen-1-yl-ben...)
Affinity DataIC50: 200nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor beta(Rat)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50225311(CHEMBL15128)
Affinity DataKd:  220nMAssay Description:Equilibrium dissociation constant for rat uterine estrogen receptor binding [3H]estradiolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2018
Entry Details Article
PubMed
TargetEstrogen receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50166895(US8552057, 4 | CHEMBL195560 | 3-(4-Hydroxy-phenyl)...)
Affinity DataIC50: 234nMAssay Description:Displacement of [3H]estradiol from rat uterine cytosolic estrogen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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