Compile Data Set for Download or QSAR
Report error Found 494 for UniProtKB: P18090
LigandPNGBDBM50497048(CHEMBL3246767)
Affinity DataIC50: 0.00130nMAssay Description:Inhibition of beta-adrenergic receptor in rat portal veinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50497052(CHEMBL3246792)
Affinity DataIC50: 0.0450nMAssay Description:Inhibition of beta-adrenergic receptor in rat portal veinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50497050(CHEMBL3244454)
Affinity DataIC50: 0.0510nMAssay Description:Inhibition of beta-adrenergic receptor in rat portal veinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor S190A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor W134A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat wild type beta-1 adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0794nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356F mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM81885(CAS_52560-77-7 | 2-(3-tert-Butylamino-2-hydroxypro...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.316nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
LigandPNGBDBM50497051(CHEMBL3246789)
Affinity DataIC50: 0.440nMAssay Description:Inhibition of beta-adrenergic receptor in rat portal veinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50497049(CHEMBL3246801)
Affinity DataIC50: 0.460nMAssay Description:Inhibition of beta-adrenergic receptor in rat portal veinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKi:  0.460nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKi:  0.610nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50019443(LB-46 | 1-(1H-Indol-4-yloxy)-3-isopropylamino-prop...)
Affinity DataKi:  0.660nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMed
LigandPNGBDBM50246936(S-(-)-propanolol | (-)-(S)-Propranolol | [2-Hydrox...)
Affinity DataKd:  0.700nMAssay Description:Binding affinity against Beta adrenergic receptor in C6-2B astrocytoma cells, using [125I]-iodohydroxybenzylpindolol-benzylpindolol([125I]-HYP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50497054(CHEMBL3246790)
Affinity DataIC50: 0.780nMAssay Description:Inhibition of beta-adrenergic receptor in rat portal veinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM25759([3-(9H-carbazol-4-yloxy)-2-hydroxypropyl][2-(2-met...)
Affinity DataKi:  0.810nMAssay Description:Displacement of [3H]CGP12177 from beta-1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50212981(CHEMBL543099 | SR-59062A)
Affinity DataIC50: 0.900nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colon in presence of phentolamine (10 uM), desmethylimipramine (0.5 uM) and hydrocortisone (30 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKd:  1nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM25764(ALPRENOLOL,(-) | CHEMBL266195 | ALPRENOLOL,(+) | A...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
LigandPNGBDBM50212980(CHEMBL553039 | SR-58997A)
Affinity DataIC50: 1.10nMAssay Description:Beta-adrenergic agonistic activity in rat proximal colon in presence of phentolamine (10 uM), desmethylimipramine (0.5 uM) and hydrocortisone (30 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKd:  1.20nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKd:  1.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50497053(CHEMBL3246795)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of beta-adrenergic receptor in rat portal veinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating beta-blo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  1.60nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating beta-blo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to membrane preparation from rat lung reticulocyte pretreated with alkylating beta-blocker...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKi:  1.80nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM25753(Artrenolol | 2-{4-[2-hydroxy-3-(propan-2-ylamino)p...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKd:  2nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding sites on beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50267197((2S)-1-(1H-Indol-4-yloxy)-3-{[2-(2-methoxyphenoxy)...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CGP12177 from beta-1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  2.10nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]Dihydroalprenolol in rat heart tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  2.40nMAssay Description:Inhibitory activity against beta adrenergic receptor of rat frontal cortex homogenate using (1.0 nM) [3H]- dihydroalprenololMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKd:  2.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  2.5nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  2.5nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  2.80nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat heart tissue at 1*10e-6 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  2.80nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-6 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKi:  2.80nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM81886(CHEMBL287651 | CAS_3506-09-0 | PROPRANOLOL, dl)
Affinity DataKi:  2.82nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50267196((+/-)1-(1H-indol-4-yloxy)-3-(2-(2-methoxyphenoxy)e...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CGP12177 from beta-1 adrenergic receptor in rat cerebral cortex by liquid scintillation methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  3nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat heart tissue at 1*10e-5 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  3nMAssay Description:Radioligand receptor binding studies were conducted in the rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2013
Entry Details Article

LigandPNGBDBM50226969(CHEMBL39915)
Affinity DataIC50: 3.10nMAssay Description:The compound was evaluated for the inhibition of [125I]cyanopindolol binding to beta adrenergic receptor in rat reticulocyte membrane.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  3.20nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]Dihydroalprenolol in rat heart tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  3.20nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]Dihydroalprenolol in rat heart tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
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