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Report error Found 106 of affinity data for UniProtKB/TrEMBL: P28838
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50367209(Ubenimex | BESTATIN HYDROCHLORIDE)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human recombinant Leucine aminopeptidase 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50277143(CHR 2797 | CHR-2797 | Tosedostat)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant Leucine aminopeptidase 3More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50017478(CHEMBL28650 | Amastatin | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  30nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50225458(CHEMBL393949 | (S)-3-[((S)-1-amino-3-phenyl-propyl...)
Affinity DataKi:  45nMAssay Description:Inhibition of pig kidney cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50457478(CHEMBL4208547)
Affinity DataKi:  50nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129685(2-Amino-4-methyl-pentanal | CHEMBL88476)
Affinity DataKi:  60nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129683(CHEMBL328319 | CHEMBL2153736 | Diastereomer-2-[(1-...)
Affinity DataKi:  65nMAssay Description:Inhibition of LAPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129683(CHEMBL328319 | CHEMBL2153736 | Diastereomer-2-[(1-...)
Affinity DataKi:  65nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129683(CHEMBL328319 | CHEMBL2153736 | Diastereomer-2-[(1-...)
Affinity DataKi:  65nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  66nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129684(3-[(1-amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  66nMAssay Description:Inhibition of pig kidney cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129681(3-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoyl]-...)
Affinity DataKi:  67nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129682(2-[(1-Amino-3-phenyl-propyl)-hydroxy-phosphinoylme...)
Affinity DataKi:  74nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50089610((Z)-(S)-5-Amino-7-methyl-4-oxo-oct-2-enoic acid me...)
Affinity DataKi:  76nMAssay Description:Inhibitory activity against leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50027041(2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-4-met...)
Affinity DataKi:  120nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 180nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50017478(CHEMBL28650 | Amastatin | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  200nMAssay Description:Effect of inhibitor structure on the slow binding inhibition of Leucine aminopeptidase was determined and the Ki was reported which is = k2/k1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50017478(CHEMBL28650 | Amastatin | Leu[1psi,CHOHCONH]ValVal...)
Affinity DataKi:  220nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50316047(1-amino-2-methylbutylphosphonic acid monophenylest...)
Affinity DataKi:  230nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129679(1-amino-3-methylbutylphosphonic acid | (1-Amino-3-...)
Affinity DataKi:  230nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50024594(LEUCINE PHOSPHONIC ACID | (R)-1-Ammonium-3-methyl-...)
Affinity DataKi:  230nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129679(1-amino-3-methylbutylphosphonic acid | (1-Amino-3-...)
Affinity DataKi:  230nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50234656(CHEMBL252204 | CHEMBL254285 | (R)-3-[((R)-1-amino-...)
Affinity DataKi:  271nMAssay Description:Inhibition of pig kidney cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 290nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 300nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129677(3-[(1-Amino-3-methyl-butyl)-hydroxy-phosphinoyl]-p...)
Affinity DataKi:  330nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50022747(CHEMBL68979 | CHEMBL304141 | 2-(3-Amino-2-hydroxy-...)
Affinity DataKi:  330nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50316048(1-amino-2-phenylethylphosphonic acid monophenyl es...)
Affinity DataKi:  420nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50024592((S)-1-Ammonium-2-phenyl-ethanephosphonic acid anio...)
Affinity DataKi:  420nMAssay Description:Inhibition of leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50024596([(1R)-1-amino-2-phenylethyl]phosphonic acid | (R)-...)
Affinity DataKi:  420nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50024590(1-Ammonium-octane-1-phosphonic acid anion | CHEMBL...)
Affinity DataKi:  470nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50027043(3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-buty...)
Affinity DataKi:  500nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase from porcine kidney and the inhibition constant was determined after preincubatin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50008431(CHEMBL309130 | 3-Amino-2-hydroxy-N-(3-methyl-butyl...)
Affinity DataKi:  510nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50022751(CHEMBL1204264 | 2-(3-Amino-2-mercapto-4-phenyl-but...)
Affinity DataKi:  550nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50027042(3-Amino-2-hydroxy-5-methyl-hexanoic acid {2-methyl...)
Affinity DataKi:  890nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50225458(CHEMBL393949 | (S)-3-[((S)-1-amino-3-phenyl-propyl...)
Affinity DataKi:  988nMAssay Description:Inhibition of pig kidney cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50024601(1-aminohexylphosphonic acid | 1-Ammonium-hexane-1-...)
Affinity DataKi:  1.00E+3nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50022751(CHEMBL1204264 | 2-(3-Amino-2-mercapto-4-phenyl-but...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50024602(1-amino-2-methylpropylphosphonic acid | 1-Ammonium...)
Affinity DataKi:  1.20E+3nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50027046(2-[2-(3-Amino-2-hydroxy-5-methyl-hexanoylamino)-3-...)
Affinity DataKi:  1.24E+3nMAssay Description:Compound was evaluated for the inhibition of Leucine aminopeptidase and the inhibition constant was determined after preincubating the enzyme and inh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50457469(CHEMBL4213478)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of LAP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50024604(1-aminopropylphosphonic acid | 1-Ammonium-propane-...)
Affinity DataKi:  3.60E+3nMAssay Description:Compound was tested for inhibition of Leucine aminopeptidase isolated from porcine kidney; Inhibitor exhibits slow-binding behavior(k on <=1000Me-1Se...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50022742(3-Amino-2-hydroxy-N-(3-methyl-butyl)-4-phenyl-thio...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50129680({[hydroxy(1-hydroxy-3-methylbutyl)phosphoryl]amino...)
Affinity DataKi:  4.88E+3nMAssay Description:Binding affinity for cytosolic leucine aminopeptidase (LAP) from porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2012
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytosol aminopeptidase(Human)TBA
LigandPNGBDBM50234656(CHEMBL252204 | CHEMBL254285 | (R)-3-[((R)-1-amino-...)
Affinity DataKi:  8.80E+3nMAssay Description:Inhibition of pig kidney cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
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