Compile Data Set for Download or QSAR
Report error Found 77 of affinity data for UniProtKB/TrEMBL: P35750
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM23865(3-[(2S)-2-[1-(9H-fluoren-9-yl)acetamido]-4-methylp...)
Affinity DataKi:  8nM ΔG°:  -45.7kJ/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2008
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50543556(CHEMBL4647187)
Affinity DataKi:  9nMAssay Description:Inhibition of mu-calpain in porcine erythrocyte using Suc-Leu-Tyr-AMC as substrate by microtiter plate assay based Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM23866(benzyl N-[(1S)-2-methyl-1-[(1-oxo-3-phenylpropan-2...)
Affinity DataKi:  10nM ΔG°:  -45.2kJ/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2008
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50014577(CHEMBL286722 | benzyl (S)-3-methyl-1-oxo-1-((S)-1-...)
Affinity DataKi:  10nMAssay Description:Inhibition of mu-calpain in porcine erythrocyte using Suc-Leu-Tyr-AMC as substrate by microtiter plate assay based Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50543555(CHEMBL4642092)
Affinity DataKi:  14nMAssay Description:Inhibition of mu-calpain in porcine erythrocyte using Suc-Leu-Tyr-AMC as substrate by microtiter plate assay based Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50543554(CHEMBL4646991)
Affinity DataKi:  16nMAssay Description:Inhibition of mu-calpain in porcine erythrocyte using Suc-Leu-Tyr-AMC as substrate by microtiter plate assay based Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50543552(CHEMBL4642290)
Affinity DataKi:  18nMAssay Description:Inhibition of mu-calpain in porcine erythrocyte using Suc-Leu-Tyr-AMC as substrate by microtiter plate assay based Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193489((R)-1-(4-nitrophenylsulfonyl)-N-((R,S)-1-oxo-3-phe...)
Affinity DataKi:  20nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326300(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  23nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193501((R)-1-(4-iodophenylsulfonyl)-N-((R,S)-1-oxo-3-phen...)
Affinity DataKi:  33nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50114340(N-(4-fluorophenylsulfonyl)-L-valyl-L-leucinal | (S...)
Affinity DataIC50: 35nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193494((R)-1-(4-methoxyphenylsulfonyl)-N-((R,S)-1-oxo-3-p...)
Affinity DataKi:  37nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326298(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  41nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM23859(3-[(2S)-2-[1-(adamantan-1-yl)acetamido]-4-methylpe...)
Affinity DataKi:  41nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2008
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193509((S)-3-(4-iodophenylsulfonyl)-N-((R,S)-1-oxo-3-phen...)
Affinity DataKi:  42nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM23857(3-[(2S)-2-(3-cyclohexylpropanamido)-4-methylpentan...)
Affinity DataKi:  50nM ΔG°:  -41.3kJ/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2008
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326303(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  53nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326304(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(6-amino-...)
Affinity DataKi:  55nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM23863(3-[(2S)-2-(3,3-diphenylpropanamido)-4-methylpentan...)
Affinity DataKi:  63nM ΔG°:  -40.7kJ/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2008
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193503((4S)-N-(1-oxo-3-phenylpropan-2-yl)-3-tosylthiazoli...)
Affinity DataKi:  70nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193502((S)-3-(4-bromophenylsulfonyl)-N-((R,S)-1-oxo-3-phe...)
Affinity DataKi:  74nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50244952((S)-2-ethyl-N-(1-oxo-3-phenylpropan-2-yl)-2-(3-phe...)
Affinity DataKi:  80nMAssay Description:Inhibition of pig erythrocyte mu-calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193507((2R)-N-(1-oxo-3-phenylpropan-2-yl)-1-tosylpyrrolid...)
Affinity DataKi:  81nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193490((S)-3-(4-chlorophenylsulfonyl)-N-((R,S)-1-oxo-3-ph...)
Affinity DataKi:  90nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM23861(3-[(2S)-2-(1,1-diphenylacetamido)-4-methylpentanam...)
Affinity DataKi:  108nM ΔG°:  -39.4kJ/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2008
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193495((S)-3-(4-fluorophenylsulfonyl)-N-((R,S)-1-oxo-3-ph...)
Affinity DataKi:  110nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193504((R)-1-(4-bromophenylsulfonyl)-N-((R,S)-1-oxo-3-phe...)
Affinity DataKi:  128nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193497((R)-1-(4-chlorophenylsulfonyl)-N-((R,S)-1-oxo-3-ph...)
Affinity DataKi:  141nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50084684({3-Methyl-1-[1-(3-morpholin-4-yl-propylaminooxalyl...)
Affinity DataKi:  150nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326299(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-amino-...)
Affinity DataKi:  165nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50069792((2S)-2-[(2S)-2-acetamido-4-methylpentanamido]-N-[(...)
Affinity DataKi:  190nMAssay Description:Inhibition of pig erythrocyte mu-calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50114336((S)-2-(4-Fluoro-benzenesulfonylamino)-N-{(S)-1-[(2...)
Affinity DataIC50: 190nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193506((R)-1-(naphthalen-1-ylsulfonyl)-N-((R,S)-1-oxo-3-p...)
Affinity DataKi:  191nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193493((R)-N-((R,S)-1-oxo-3-phenylpropan-2-yl)-1-(phenyls...)
Affinity DataKi:  196nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326306(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(dimethyl...)
Affinity DataKi:  226nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193505((R)-1-(3-nitrophenylsulfonyl)-N-((R,S)-1-oxo-3-phe...)
Affinity DataKi:  256nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50543553(CHEMBL4640485)
Affinity DataKi:  273nMAssay Description:Inhibition of mu-calpain in porcine erythrocyte using Suc-Leu-Tyr-AMC as substrate by microtiter plate assay based Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193500((R)-N-(2(R,S)-3,4-dioxo-4-(phenethylamino)-1-pheny...)
Affinity DataKi:  280nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193499((R)-1-(butylsulfonyl)-N-((R,S)-1-oxo-3-phenylpropa...)
Affinity DataKi:  313nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50114342((S)-N-{(S)-1-[(2-Dimethylamino-acetyl)-hydrazonome...)
Affinity DataIC50: 370nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193496((R)-1-(4-fluorophenylsulfonyl)-N-((R,S)-1-oxo-3-ph...)
Affinity DataKi:  386nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193508((R)-1-(2-nitrophenylsulfonyl)-N-((R,S)-1-oxo-3-phe...)
Affinity DataKi:  424nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193492((R)-N-(2(R,S)-3,4-dioxo-4-(phenethylamino)-1-pheny...)
Affinity DataKi:  450nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM23858(methyl 3-[(2S)-2-[1-(adamantan-1-yl)acetamido]-4-m...)
Affinity DataKi:  450nM ΔG°:  -35.9kJ/molepH: 7.4 T: 2°CAssay Description:Assays were initiated by addition of CaCl2, and the increase in fluorescence (ex @370 nm, em @440 nm) was monitored. MDL28170 and buffer with 2% DMSO...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2008
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326301(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-amino-...)
Affinity DataKi:  480nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326302(3-(Benzyloxycarbonyl-L-leucylamino)-N-(3-(4-methyl...)
Affinity DataKi:  640nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50114341((2S)-N-((1S)-1-{(E)-[(aminocarbonyl)hydrazono]meth...)
Affinity DataIC50: 680nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50326305(3-(Benzyloxycarbonyl-L-leucylamino)-N-(2-(dimethyl...)
Affinity DataKi:  711nMAssay Description:Inhibition of porcine erythrocyte calpain 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2011
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50114337((S)-2-(4-Fluoro-benzenesulfonylamino)-3-methyl-N-{...)
Affinity DataIC50: 790nMAssay Description:Tested for inhibitory activity against porcine erythrocyte Mu-calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCalpain-1 catalytic subunit(Pig)
University of Tennessee Health Science Center

LigandPNGBDBM50193498((R)-1-(isopropylsulfonyl)-N-((R,S)-1-oxo-3-phenylp...)
Affinity DataKi:  836nMAssay Description:Inhibition of porcine erythrocyte mu calpainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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