Compile Data Set for Download or QSAR
Report error Found 130 of affinity data for UniProtKB/TrEMBL: Q64610
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699087BDBM699087(4-(8-((2-fluoro-5-(trifluoromethyl)benzoyl)-D- val...)
Affinity DataIC50: 1.10nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285776BDBM50285776(CHEMBL4172309)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285750BDBM50285750(CHEMBL4173049)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699076BDBM699076(2-fluoro-N-((2R)-1-(4-(4-methoxyphenyl)-2- methyl-...)
Affinity DataIC50: 1.70nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285745BDBM50285745(CHEMBL4162641)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285744BDBM50285744(CHEMBL4168498)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699090BDBM699090(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-4-(p- tolyl)...)
Affinity DataIC50: 2.20nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285774BDBM50285774(CHEMBL4169550)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285748BDBM50285748(CHEMBL4173341)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285751BDBM50285751(CHEMBL4169912)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285777BDBM50285777(CHEMBL4165749 | BI-2545 (19))
Affinity DataIC50: 3.40nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699084BDBM699084(N-((2R)-1-(4-(4-fluorophenyl)-2-methyl-2,8- diazas...)
Affinity DataIC50: 3.40nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699100BDBM699100(2-fluoro-N-((2R)-3-methyl-1-oxo-1-(10-oxo-7- pheny...)
Affinity DataIC50: 3.5nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699072BDBM699072(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-1-oxo-4- phe...)
Affinity DataIC50: 3.80nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699056BDBM699056(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-1-oxo-4- phe...)
Affinity DataIC50: 4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699094BDBM699094(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- methyl-2...)
Affinity DataIC50: 4.10nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699093BDBM699093(N-((1R)-1-cyclohexyl-2-(4-(4-fluorophenyl)-2- meth...)
Affinity DataIC50: 4.40nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285774BDBM50285774(CHEMBL4169550)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of ATX in rat whole blood using LPA 17:0 as substrate after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285773BDBM50285773(CHEMBL4170966)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699108BDBM699108(2-fluoro-N-((2R)-1-(7-(4-fluorophenyl)-9- methyl-3...)
Affinity DataIC50: 5.10nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285743BDBM50285743(CHEMBL4169136)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699101BDBM699101(2-fluoro-N-((2R)-1-(7-(4-fluorophenyl)-10-oxo- 3,9...)
Affinity DataIC50: 6.5nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699061BDBM699061(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-4- phenyl-2,...)
Affinity DataIC50: 6.60nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699082BDBM699082(2-fluoro-N-((2R)-1-(4-(4-methoxyphenyl)-2- methyl-...)
Affinity DataIC50: 6.80nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699065BDBM699065(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- methyl-1...)
Affinity DataIC50: 6.90nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699063BDBM699063(N-((2R)-1-(4-(1H-indazol-5-yl)-2-methyl-2,8- diaza...)
Affinity DataIC50: 6.90nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285775BDBM50285775(CHEMBL4159308)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of ATX in rat whole blood using LPA 17:0 as substrate after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699098BDBM699098(N-((2R)-1-(4-(4-fluorophenyl)-2-methyl-2,8- diazas...)
Affinity DataIC50: 6.90nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285748BDBM50285748(CHEMBL4173341)
Affinity DataIC50: 7nMAssay Description:Inhibition of ATX in rat whole blood using LPA 17:0 as substrate after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699079BDBM699079(2-fluoro-N-((2R)-1-(4-(4-fluorophenyl)-2- methyl-2...)
Affinity DataIC50: 7.10nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699103BDBM699103(2-fluoro-N-((2R)-1-(7-(4-fluorophenyl)-9- methyl-1...)
Affinity DataIC50: 7.5nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699089BDBM699089(2-fluoro-N-((R)-1-((S)-4-(4-fluorophenyl)-2- methy...)
Affinity DataIC50: 7.80nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50605406BDBM50605406(CHEMBL5190935)
Affinity DataKi:  9nMAssay Description:Inhibition of rat ATX by Michaelis-Menten analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699083BDBM699083(2-fluoro-N-((2R)-1-(4-(4-methoxyphenyl)-2- methyl-...)
Affinity DataIC50: 9.30nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699107BDBM699107(2-fluoro-N-((2R)-3-methyl-1-(9-methyl-7- phenyl-3,...)
Affinity DataIC50: 9.90nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285778BDBM50285778(CHEMBL4164935)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699071BDBM699071(2-fluoro-5-methyl-N-((2R)-3-methyl-1-(2- methyl-1-...)
Affinity DataIC50: 10.1nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699099BDBM699099(4-methyl-N-((2R)-3-methyl-1-(2-methyl-4- (pyridin-...)
Affinity DataIC50: 10.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699102BDBM699102(2-fluoro-N-((2R)-3-methyl-1-(9-methyl-10-oxo- 7-ph...)
Affinity DataIC50: 11.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699092BDBM699092(2-fluoro-N-((1R)-2-(4-(4-fluorophenyl)-2- methyl-2...)
Affinity DataIC50: 11.5nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699066BDBM699066(N-((2R)-1-(2-ethyl-4-(4-fluorophenyl)-1-oxo-2,8- d...)
Affinity DataIC50: 11.7nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699088BDBM699088(2-fluoro-N-((R)-1-((R)-4-(4-fluorophenyl)-2- methy...)
Affinity DataIC50: 12nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699105BDBM699105(2-fluoro-N-((2S)-3-methyl-1-(9-methyl-10-oxo- 7-ph...)
Affinity DataIC50: 12nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699058BDBM699058(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-1-oxo-4- (py...)
Affinity DataIC50: 13.3nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699062BDBM699062(2-fluoro-N-((2R)-3-methyl-1-(2-methyl-4- (pyridin-...)
Affinity DataIC50: 13.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285742BDBM50285742(CHEMBL4163050)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant rat ATX using LPC 18:1 as substrate after 2 hrs by rapidfire/MS-based analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699106BDBM699106(N-((2R)-3-methyl-1-(9-methyl-10-oxo-7-phenyl- 3,9-...)
Affinity DataIC50: 15.9nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699070BDBM699070(N-((2R)-3-methyl-1-(2-methyl-1-oxo-4-phenyl- 2,8-d...)
Affinity DataIC50: 16.4nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 699104BDBM699104(N-((2R)-1-(9-ethyl-7-(4-fluorophenyl)-10-oxo- 3,9-...)
Affinity DataIC50: 17.2nMAssay Description:The biochemical reaction consisted of 50 mM Tris (pH 8.0), 3 mM KCl, 1 mM CaCl2, 1 mM Mg Cl2, 0.14 mM NaCl and 0.1% bovine serum albumin, which was s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2025
Entry Details
US Patent

TargetAutotaxin(Rat)
Zydus Lifesciences

US Patent
LigandChemical structure of BindingDB Monomer ID 50285750BDBM50285750(CHEMBL4173049)
Affinity DataIC50: 18nMAssay Description:Inhibition of ATX in rat whole blood using LPA 17:0 as substrate after 1 hr by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
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