Compile Data Set for Download or QSAR
Report error Found 241 of affinity data for UniProtKB/TrEMBL: Q6TY19
TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379670BDBM379670(US9926281, Compound 194 | US9926281, Compound 413)
Affinity DataIC50: 5nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379686BDBM379686(US9926281, Compound 212)
Affinity DataIC50: 5nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379681BDBM379681(US9926281, Compound 416 | US9926281, Compound 207)
Affinity DataIC50: 6nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379668BDBM379668(US9926281, Compound 192 | US9926281, Compound 411)
Affinity DataIC50: 6nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379653BDBM379653(US9926281, Compound 176)
Affinity DataIC50: 7nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379669BDBM379669(US9926281, Compound 193 | US9926281, Compound 412)
Affinity DataIC50: 7nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379645BDBM379645(US9926281, Compound 408 | US9926281, Compound 167)
Affinity DataIC50: 10nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379649BDBM379649(US9926281, Compound 172 | US9926281, Compound 409)
Affinity DataIC50: 11nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379678BDBM379678(US9926281, Compound 204)
Affinity DataIC50: 11nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379667BDBM379667(US9926281, Compound 191)
Affinity DataIC50: 11nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 471764BDBM471764((5S)-5- cyclopropyl- 5-[(2S)-3-[4-(3- fluoro-5-met...)
Affinity DataIC50: 12.5nMAssay Description:TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 471793BDBM471793(5-[3-[(3S)-4-(3,4- difluoro-5- methoxy-phenyl)- 3-...)
Affinity DataIC50: 12.5nMAssay Description:TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 471794BDBM471794(5-[3-[4-(3,4- difluoro-5- methoxy- phenyl) piperaz...)
Affinity DataIC50: 12.5nMAssay Description:TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 471743BDBM471743(5-cyclopropyl-5- [3-[(3S)-4-(3,4- difluoro-5- meth...)
Affinity DataIC50: 12.5nMAssay Description:TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 429696BDBM429696(US10550100, Compound 29 | 5-(3-(4-(3- chlorophenyl...)
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H).For the d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 471792BDBM471792(5-[3-[4-(4-chloro- 3-methoxy- phenyl)-3-methyl- pi...)
Affinity DataIC50: 12.5nMAssay Description:TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 471788BDBM471788((5S)-5- cyclopropyl- 5-[3-[(3S)-4-(3,4- difluoro-5...)
Affinity DataIC50: 12.5nMAssay Description:TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 429695BDBM429695(US10550100, Compound 28 | 5-(3-(4-(3- fluorophenyl...)
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H).For the d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 471834BDBM471834((5S)-5-[(2S)-3-[4- (3,4-difluoro-5- methoxy- pheny...)
Affinity DataIC50: 12.5nMAssay Description:TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 471828BDBM471828((5S)-5-[(2S)-3-[4- (3,4-difluoro-5- methoxy- pheny...)
Affinity DataIC50: 12.5nMAssay Description:TABLE VII: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID NO: 2) by rnADAMTS-5 (1-564-6H...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/28/2021
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379666BDBM379666(US9926281, Compound 190)
Affinity DataIC50: 15nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379692BDBM379692(US9926281, Compound 218)
Affinity DataIC50: 17nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379651BDBM379651(US9926281, Compound 174)
Affinity DataIC50: 17nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379689BDBM379689(US9926281, Compound 215)
Affinity DataIC50: 18nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379703BDBM379703(US9926281, Compound 405 | US9926281, Compound 422)
Affinity DataIC50: 18nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379704BDBM379704(US9926281, Compound 432 | US9926281, Compound 406)
Affinity DataIC50: 20nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379694BDBM379694(US9926281, Compound 233)
Affinity DataIC50: 20nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379673BDBM379673(US9926281, Compound 197)
Affinity DataIC50: 21nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379687BDBM379687(US9926281, Compound 213)
Affinity DataIC50: 21nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379650BDBM379650(US9926281, Compound 173)
Affinity DataIC50: 21nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379652BDBM379652(US9926281, Compound 175)
Affinity DataIC50: 22nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379698BDBM379698(US9926281, Compound 265)
Affinity DataIC50: 22nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379697BDBM379697(US9926281, Compound 255)
Affinity DataIC50: 23nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379685BDBM379685(US9926281, Compound 211)
Affinity DataIC50: 23nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379606BDBM379606(US9926281, Compound 103)
Affinity DataIC50: 24nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379620BDBM379620(US9926281, Compound 121)
Affinity DataIC50: 24nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379677BDBM379677(US9926281, Compound 203)
Affinity DataIC50: 26nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379647BDBM379647(US9926281, Compound 169)
Affinity DataIC50: 27nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379679BDBM379679(US9926281, Compound 205)
Affinity DataIC50: 27nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379676BDBM379676(US9926281, Compound 200 | US9926281, Compound 219)
Affinity DataIC50: 29nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379557BDBM379557(US9926281, Compound 36)
Affinity DataIC50: 29nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379619BDBM379619(US9926281, Compound 116)
Affinity DataIC50: 29nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379688BDBM379688(US9926281, Compound 214)
Affinity DataIC50: 30nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379656BDBM379656(US9926281, Compound 179)
Affinity DataIC50: 34nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379696BDBM379696(US9926281, Compound 249)
Affinity DataIC50: 34nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379701BDBM379701(US9926281, Compound 314)
Affinity DataIC50: 34nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379641BDBM379641(US9926281, Compound 160)
Affinity DataIC50: 36nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379565BDBM379565(US9926281, Compound 55)
Affinity DataIC50: 37nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379642BDBM379642(US9926281, Compound 161)
Affinity DataIC50: 37nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

TargetADAMTS5(Rat)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 379621BDBM379621(US9926281, Compound 124)
Affinity DataIC50: 37nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details
US Patent

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