Compile Data Set for Download or QSAR
Report error Found 13 of affinity data for UniProtKB/TrEMBL: Q8IBS5
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50530637(CHEMBL4591417)
Affinity DataKd:  50nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50530637(CHEMBL4591417)
Affinity DataKd:  50nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50530637(CHEMBL4591417)
Affinity DataKd:  50nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50530659(CHEMBL4461850)
Affinity DataKd:  60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50530659(CHEMBL4461850)
Affinity DataKd:  60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50530659(CHEMBL4461850)
Affinity DataKd:  60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr in presence of ATP-competitive kinase inhibitor by kino...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50530637(CHEMBL4591417)
Affinity DataKd:  50nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50530659(CHEMBL4461850)
Affinity DataKd:  60nMAssay Description:Binding affinity to CDPK4 in Plasmodium falciparum 3D7 blood stage extract incubated for 1 hr by kinobeads based pull down assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383381(CHEMBL2070050 | CHEMBL2030554 | US9765037, Compoun...)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDPK4 in Plasmodium falciparum 3D7 microgametesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50383381(CHEMBL2070050 | CHEMBL2030554 | US9765037, Compoun...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Plasmodium falciparum CDPK4 using syntide-2 as substrate by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50389704(CHEMBL2070081 | US9518026, Example 9 | US9765037, ...)
Affinity DataIC50: 10nMAssay Description:Inhibition of Plasmodium falciparum CDPK4 using syntide-2 as substrate by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50345704(CHEMBL1231371 | CHEMBL2069957 | 1-(tert-butyl)-3-(...)
Affinity DataIC50: 177nMAssay Description:Inhibition of CDPK4 in Plasmodium falciparum 3D7 microgametesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCalcium-dependent protein kinase 4(Plasmodium falciparum (isolate 3D7))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM79181(cid_2913535 | TRIFLUOPERAZINE | SMR000059133 | MLS...)
Affinity DataKi:  1.50E+5nMAssay Description:Inhibition of Plasmodium falciparum His-tagged CDPK4 expressed in Escherichia coli BL21(DE3) using EGTA as substrate after 10 mins in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed