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11 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of 4-(Arylethynyl)piperidine Derivatives as Potent Nonsaccharide O-GlcNAcase Inhibitors for the Treatment of Alzheimer's Disease.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Design, synthesis and evaluation of novel UDCA-aminopyrimidine hybrids as ATX inhibitors for the treatment of hepatic and pulmonary fibrosis.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Design, synthesis and biological evaluation of biaryl amide derivatives against SARS-CoV-2 with dual-target mechanism.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Discovery of 2-Ethoxy-5-isobutyramido-N-1-substituted Benzamide Derivatives as Selective Kv2.1 Inhibitors with In Vivo Neuroprotective Effects.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Discovery of Natural Ah Receptor Antagonists from Salvia miltiorrhiza Bunge and Synthesis of Analogs for Tumor Immunotherapy.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Design, Synthesis, and Bioevaluation of Novel Reversibly Photoswitchable PI3K Inhibitors Based on Phenylazopyridine Derivatives toward Light-Controlled Cancer Treatment.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Discovery of Oral AMP-Activated Protein Kinase Activators for Treating Hyperlipidemia.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Discovery of ganoderic acid A (GAA) PROTACs as MDM2 protein degraders for the treatment of breast cancer.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Discovery of Quinazoline-2,4(1EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Discovery of a Novel Photocaged PI3K Inhibitor Capable of Real-Time Reporting of Drug Release.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College
Synthesis and structure-activity relationships of N - (3 - (1H-imidazol-2-yl) phenyl) - 3-phenylpropionamide derivatives as a novel class of covalent inhibitors of p97/VCP ATPase.EBI
Chinese Academy of Medical Sciences and Peking Union Medical College