16 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
Organization
Discovery of Highly Selective Inhibitors of the Immunoproteasome Low Molecular Mass Polypeptide 2 (LMP2) Subunit.
Kezar Life Sciences
Structure-based design of฿1i or฿5i specific inhibitors of human immunoproteasomes.
Leiden Institute of Chemistry and Netherlands Proteomics Centre
Identification of N, C-capped di- and tripeptides as selective immunoproteasome inhibitors.
Chinese Academy of Medical Sciences and Peking Union Medical College
Structure-Based Optimization and Discovery of M3258, a Specific Inhibitor of the Immunoproteasome Subunit LMP7 (?5i).
Merck
Cell-based screening of extracts of natural sources to search for inhibitors of the ubiquitin-proteasome system and identification of proteasome inhibitors from the fungus Remotididymella sp.
Kumamoto University
Development of peptide epoxyketones as selective immunoproteasome inhibitors.
Zhejiang University
Macrocyclic Immunoproteasome Inhibitors as a Potential Therapy for Alzheimer's Disease.
University of Kentucky
Target Validation and Identification of Novel Boronate Inhibitors of the Plasmodium falciparum Proteasome.
The University of Melbourne
LMP2 Inhibitors as a Potential Treatment for Alzheimer's Disease.
University of Kentucky
Exploration of novel macrocyclic dipeptide N-benzyl amides as proteasome inhibitors.
Zhejiang University
Required Immunoproteasome Subunit Inhibition Profile for Anti-Inflammatory Efficacy and Clinical Candidate KZR-616 ((2 S,3 R)- N-(( S)-3-(Cyclopent-1-en-1-yl)-1-(( R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-hydroxy-3-(4-methoxyphenyl)-2-(( S)-2-(2-morpholinoacetamido)propanamido)propenamide).
Kezar Life Sciences
Immunoproteasome-selective inhibitors: An overview of recent developments as potential drugs for hematologic malignancies and autoimmune diseases.
Hangzhou Xixi Hospital
Development of Novel Epoxyketone-Based Proteasome Inhibitors as a Strategy To Overcome Cancer Resistance to Carfilzomib and Bortezomib.
University of Kentucky
Structure-Based Design of Inhibitors Selective for Human Proteasome ?2c or ?2i Subunits.
Leiden Institute of Chemistry and Netherlands Proteomics Centre
Tetradehydrohalicyclamine B, a new proteasome inhibitor from the marine sponge Acanthostrongylophora ingens.
Kumamoto University