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26 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Design and synthesis of selective, dual fatty acid binding protein 4 and 5 inhibitors.EBI
F. Hoffmann-La Roche
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation.EBI
Chinese Academy of Sciences
Interaction Analysis of FABP4 Inhibitors by X-ray Crystallography and Fragment Molecular Orbital Analysis.EBI
Ajinomoto
Novel fatty acid binding protein 4 (FABP4) inhibitors: virtual screening, synthesis and crystal structure determination.EBI
Chinese Academy of Sciences
Structure-guided design, synthesis and in vitro evaluation of a series of pyrazole-based fatty acid binding protein (FABP) 3 ligands.EBI
Okayama University 1-1-1
Simple, intuitive calculations of free energy of binding for protein-ligand complexes. 1. Models without explicit constrained water.EBI
University of Parma
New aromatic substituted pyrazoles as selective inhibitors of human adipocyte fatty acid-binding protein.EBI
Chinese Academy of Sciences
Discovery of highly selective inhibitors of human fatty acid binding protein 4 (FABP4) by virtual screening.EBI
Chinese Academy of Sciences
Identification and characterization of a small molecule inhibitor of Fatty Acid binding proteins.EBI
University of Minnesota
N-Benzyl-indolo carboxylic acids: Design and synthesis of potent and selective adipocyte fatty-acid binding protein (A-FABP) inhibitors.EBI
Biovitrum
Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP).EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
NMR structure of a potent small molecule inhibitor bound to human keratinocyte fatty acid-binding protein.EBI
Bristol-Myers Squibb Pharmaceutical Research Institute
Fragment-to-Lead Medicinal Chemistry Publications in 2020.EBI
Vrije Universiteit Amsterdam
Adipocyte fatty acid binding protein 4 (FABP4) inhibitors. An update from 2017 to early 2022.EBI
Universit£
Substituted benzylamino-6-(trifluoromethyl)pyrimidin-4(1H)-ones: a novel class of selective human A-FABP inhibitors.EBI
Biovitrum
Discovery of inhibitors of human adipocyte fatty acid-binding protein, a potential type 2 diabetes target.EBI
Biovitrum
Development of FABP4/5 inhibitors with potential therapeutic effect on type 2 Diabetes Mellitus.EBI
Fudan University
Exploration of Fragment Binding Poses Leading to Efficient Discovery of Highly Potent and Orally Effective Inhibitors of FABP4 for Anti-inflammation.EBI
Chinese Academy of Sciences
1,2,4-Triazolo[1,5-a]pyrimidines in drug design.EBI
University of California
Identification of new dual FABP4/5 inhibitors based on a naphthalene-1-sulfonamide FABP4 inhibitor.EBI
Fudan University
From hit to lead: Structure-based discovery of naphthalene-1-sulfonamide derivatives as potent and selective inhibitors of fatty acid binding protein 4.EBI
Fudan University
Synthesis and structure based optimization of novel Akt inhibitors.BDB
Pfizer
Inhibition of Src kinase activity by 4-anilino-7-thienyl-3-quinolinecarbonitriles.BDB
Wyeth Research