Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 787
LigandChemical structure of BindingDB Monomer ID 4552BDBM4552(CHEMBL288441 | SKI-606 | 4-[(2,4-Dichloro-5-methox...)
Affinity DataIC50: 1.20nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 6113BDBM6113(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-{5-[(4-h...)
Affinity DataIC50: 1.40nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6115BDBM6115(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-{5-[(4-h...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6108BDBM6108(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-[5-(morp...)
Affinity DataIC50: 2.5nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6107BDBM6107(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-[5-(morp...)
Affinity DataIC50: 2.70nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6112BDBM6112(3-quinolinecarbonitrile analog 2a | 4-[(2,4-dichlo...)
Affinity DataIC50: 3.80nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6114BDBM6114(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-{5-[(4-m...)
Affinity DataIC50: 3.80nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6116BDBM6116(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-[5-(pipe...)
Affinity DataIC50: 4.20nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6117BDBM6117(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-[5-(thio...)
Affinity DataIC50: 4.40nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6109BDBM6109(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-[4-(morp...)
Affinity DataIC50: 5.70nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6111BDBM6111(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-[4-(morp...)
Affinity DataIC50: 240nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6118BDBM6118(4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-[5-(morp...)
Affinity DataIC50: 280nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 6110BDBM6110(4-[(2,4-dichloro-5-methoxyphenyl)amino]-7-[2-(morp...)
Affinity DataIC50: 440nMpH: 7.5 T: 2°CAssay Description:Src kinase activity was measured in an ELISA format. IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2005
Entry Details Article
PubMed