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BindingDB contains 3.2M data for 1.4M Compounds and 11.5K Targets. Of those, 1.6M data for 765K Compounds and 4.8K Targets were curated by BindingDB curators. BindingDB is a FAIRsharing resource.

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21 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Cmpds
Data
Article Title
Organization
20
An insight on synthetic and medicinal aspects of pyrazolo[1,5-a]pyrimidine scaffold.EBI
University of Kwazulu-Natal
39
Ion channels as therapeutic targets: a drug discovery perspective.EBI
Pfizer
44
Selective influence on contextual memory: physiochemical properties associated with selectivity of benzodiazepine ligands at GABAA receptors containing the alpha5 subunit.EBI
Moltech
3
Azaflavones compared to flavones as ligands to the benzodiazepine binding site of brain GABA(A) receptors.EBI
Lund University
7
Synthesis of GABAA receptor agonists and evaluation of their alpha-subunit selectivity and orientation in the GABA binding site.EBI
Johannes Gutenberg University
14
Advances in Epilepsy: Mechanisms, Clinical Trials, and Drug Therapies.EBI
Sichuan University
21
A Molecular Toolbox of Positron Emission Tomography Tracers for General Anesthesia Mechanism Research.EBI
Xiamen University
173
β-Carboline as a Privileged Scaffold for Multitarget Strategies in Alzheimer's Disease Therapy.EBI
Univ. Grenoble Alpes
3
Pharmacological Analysis of the Anti-inflammatory and Antiallodynic Effects of Zinagrandinolide E from EBI
Universidad Nacional Aut£Noma De M£Xico
32
Synthesis and biological evaluation of 7,8,9,10-tetrahydroimidazo[1,2-c]pyrido[3,4-e]pyrimdin-5(6H)-ones as functionally selective ligands of the benzodiazepine receptor site on the GABA(A) receptor.EBI
Neurogen
56
Imidazopyridine-based selective and multifunctional ligands of biological targets associated with psychiatric and neurodegenerative diseases.EBI
Palack£
32
Subtype Selective γ-Aminobutyric Acid Type A Receptor (GABAEBI
University of Sussex
1
SALT AND CRYSTAL FORM OF DIPEPTIDYL PEPTIDASE INHIBITOR COMPOUNDBDB
Haisco Pharmaceuticals
80
Pyridine derivativesBDB
Astellas Pharma
80
Aromatic heterocyclic compoundBDB
Mitsubishi Tanabe Pharma
44
Factor XIa inhibitorsBDB
Merck Sharp & Dohme
166
Compounds, compositions, and methodsBDB
Denali Therapeutics
28
Design of isoform-selective phospholipase D inhibitors that modulate cancer cell invasiveness.BDB
Vanderbilt University
84
Discovery and structure-activity relationship analysis of Staphylococcus aureus sortase A inhibitors.BDB
University of California Los Angeles
21
Identification of 2-aminobenzimidazoles as potent melanin-concentrating hormone 1-receptor (MCH1R) antagonists.BDB
Banyu Pharmaceutical
54
Synthesis and SAR of tolylamine 5-HT6 antagonists.BDB
Pfizer