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30 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Development of new Malt1 inhibitors and probes.EBI
Leiden University
MALT1 Inhibitors May Potentially Treat Lymphomas and Autoimmune Disorders.EBI
Therachem Research Medilab (India)
Identification ofß-Lapachone Analogs as Novel MALT1 Inhibitors To Treat an Aggressive Subtype of Diffuse Large B-Cell Lymphoma.EBI
Institute of Basic Science (Ibs)
The Inhibitors of Mucosa-Associated Lymphoid Tissue Lymphoma Translocation Protein 1 (MALT-1) Protease as Potential Treatment of ABC-DLBCL and Similar Diseases.EBI
PI Health Sciences
Development of Potent MALT1 Inhibitors Featuring a Novel "2-Thioxo-2,3-dihydrothiazolo[4,5-d]pyrimidin-7(6H)-one" Scaffold for the Treatment of B Cell Lymphoma.EBI
Shanghai Institute of Materia Medica
Discovery of orally bioavailable inhibitors of MALT1 with in vivo activity for psoriasis.EBI
Toray Industries
Discovery and optimization of cyclohexane-1,4-diamines as allosteric MALT1 inhibitors.EBI
Astrazeneca
Identification of Novel Fused Heteroaromatics-Based MALT1 Inhibitors by High-Throughput Screening to Treat B Cell Lymphoma.EBI
Chinese Academy of Sciences
Structure-activity relationship studies of 3-substituted pyrazoles as novel allosteric inhibitors of MALT1 protease.EBI
Toray Industries
Optimization of the EBI
Novartis Pharma
Discovery of Potent, Highly Selective, and EBI
Novartis Institutes For Biomedical Research
Quinoline and thiazolopyridine allosteric inhibitors of MALT1.EBI
Harvard Medical School
Secondary Metabolites from the Fungus Dictyosporium sp. and Their MALT1 Inhibitory Activities.EBI
National Cancer Institute
Discovery and optimization of a series of small-molecule allosteric inhibitors of MALT1 protease.EBI
Janssen Research & Development
Use of Non-Natural Amino Acids for the Design and Synthesis of a Selective, Cell-Permeable MALT1 Activity-Based Probe.EBI
Ku Leuven
Peptide-based covalent inhibitors of MALT1 paracaspase.EBI
Harvard Medical School
N-aryl-piperidine-4-carboxamides as a novel class of potent inhibitors of MALT1 proteolytic activity.EBI
Novartis Institutes For Biomedical Research
Derivatives of adamantyl oxadiazoles and pharmaceutically acceptable solvates, hydrates and salts thereof, pharmaceutical composition comprising same, synthesis method, suitable for use as effective and selective inhibitors of the reductase activity of the enzyme 11-beta dehydrogenase type 1)BDB
Pontificia Universidad Catolica De Chile
DUAL-TARGETED RNA POLYMERASE INHIBITORS: CONJUGATES OF BENZOXAZINO- AND SPIRO-RIFAMYCINS WITH N ALPHA-AROYL-N-ARYL-PHENYLALANINAMIDESBDB
The State University of New Jersey
HETEROCYCLE-CONTAINING LONP1 INHIBITOR COMPOUNDS, USES AND METHODSBDB
Pretzel Therapeutics
Substituted pyrazolo[5′,1′:2,3]pyrimido[5,4-b][1,4]oxazines as TYK2 inhibitorsBDB
Takeda Pharmaceutical
N6-ADENOSINE-METHYLTRANSFERASE INHIBITORS IN CANCER TREATMENTBDB
University of Zurich
MODULATORS OF PROGRAMMED DEATH-LIGAND-1BDB
Southern Research Institute
Compounds useful as inhibitors of isoprenylcysteine carboxyl methyltransferaseBDB
Agency For Science, Technology and Research
ORALLY BIOAVAILABLE, BRAIN-PENETRANT COMPOUND WITH SELECTIVITY FOR THE CANNABINOID TYPE 2 RECEPTOR WITH POTENTIAL USE TOWARDS VISCERAL PAIN MANAGEMENT AND NEURODEGENERATIVE DISORDERSBDB
University of Mississippi
Heteroaryl compounds and their use as therapeutic drugsBDB
Dong-A Socio Holdings
Pyridazinones as PARP7 inhibitorsBDB
Ribon Therapeutics
Small-molecule HSP90 inhibitorsBDB
Sloan-Kettering Institute For Cancer Research
 
Inhibition of SARS-CoV-2 main protease by allosteric drug-bindingBDB
Center For Free-Electron Laser Science
Tropomyosin-related kinase inhibitorsBDB
Pfizer